SCHEMBL6211397

SCHEMBL6211397

CC(CCNC(=O)c1ccc(-c2ncc[nH]2)cc1)CC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.35
LMNA P02545 2/20 0.35
MAPK14 Q16539 1/20 0.34
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
CHRM4 P08173 1/20 0.33
ALDH1A1 P00352 2/20 0.32
PTAFR P25105 2/20 0.32
HTT P42858 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
F10 P00742 2/20 0.31
PRSS1 P07477 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211238 0.90 MAPK14 (0.35) SMYD3LMNAMAPK14DRD2DRD3
SCHEMBL6208718 0.88 LMNA (0.42) SMYD3LMNACHRM4ALDH1A1HTT
SCHEMBL6209450 0.87 CXCR3 (0.43) SMYD3LMNACHRM4PTAFRHPGD
SCHEMBL6211038 0.87 CTSK (0.41) SMYD3LMNAALDH1A1HTTNPSR1
SCHEMBL6211570 0.87 SLC6A5 (0.38) SMYD3LMNACHRM4
SCHEMBL6210230 0.87 ROCK2 (0.40) SMYD3LMNAALDH1A1PTAFR
SCHEMBL6210489 0.87 CHRM4 (0.39) SMYD3LMNADRD2CHRM4
SCHEMBL6212884 0.86 LMNA (0.37) SMYD3LMNACHRM4ALDH1A1HTT
SCHEMBL6209295 0.86 CTSK (0.37) SMYD3LMNADRD3ALDH1A1
SCHEMBL6213867 0.86 CHRM4 (0.40) SMYD3LMNACHRM4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed