SCHEMBL6354293

SCHEMBL6354293

Cc1cc(Cl)cc(C)c1CBr

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
RAPGEF4 Q8WZA2 2/20 0.34
SCN4A P35499 4/20 0.34
CES1 P23141 1/20 0.32
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6355236 0.88 RAPGEF4 (0.39) TSHRRAPGEF4SCN4ACYP3A4MAPT
SCHEMBL25247894 0.84 SCN4A (0.30) RAPGEF4SCN4A
SCHEMBL21803257 0.84 SCN4A (0.30) SCN4A
SCHEMBL585059 0.78 HRH3 (0.40) TSHRRAPGEF4MAPT
SCHEMBL893003 0.78 ALDH1A1 (0.41) TSHRCYP3A4
SCHEMBL21749452 0.76 HTR1D (0.41)
SCHEMBL21472699 0.76 RAPGEF4 (0.40) TSHRRAPGEF4SCN4ACES1CYP3A4
SCHEMBL14524295 0.76 TSHR (0.37) TSHRRAPGEF4SCN4ACES1CYP3A4
SCHEMBL16670956 0.76 TRPA1 (0.33) TSHR
SCHEMBL17648045 0.76 HRH3 (0.39) TSHRRAPGEF4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3774719-B1 METHOD FOR THE PREPARATION OF 2.6-DIALKYLPHENYL ACETIC ACIDS BAYER AG (DE) 2025-07-23 EP disclosed
US-20240002344-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR HISTONE LYSINE DEMETHYLASE INHIBITION FIBROGEN, INC. 2024-01-04 US disclosed
EP-4204400-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR HISTONE LYSINE DEMETHYLASE INHIBITION Fibrogen, Inc. (US) 2023-07-05 EP disclosed
US-11691938-B2 Process for preparing 2,6-dialkylphenylacetic acids BAYER AKTIENGESELLSCHAFT (DE) 2023-07-04 US disclosed
US-11691938-B2 Process for preparing 2,6-dialkylphenylacetic acids BAYER AKTIENGESELLSCHAFT (DE) 2023-07-04 US disclosed
CN-116348450-A Compounds, compositions and methods for histone lysine demethylase inhibition 菲布罗根有限公司 2023-06-27 CN disclosed
WO-2022047230-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR HISTONE LYSINE DEMETHYLASE INHIBITION FIBROGEN, INC. (US) 2022-03-03 WO disclosed
US-20210403406-A1 PROCESS FOR PREPARING 2,6-DIALKYLPHENYLACETIC ACIDS BAYER AKTIENGESELLSCHAFT (DE) 2021-12-30 US disclosed
CN-112004795-A Process for preparing 2, 6-dialkylphenylacetic acid 拜耳公司 2020-11-27 CN disclosed
WO-2019197232-A1 PROCESS FOR PRODUCING 2,6-DIALKYLPHENYL ACETIC ACIDS BAYER AKTIENGESELLSCHAFT (DE) 2019-10-17 WO disclosed
US-20030220364-A1 New compounds AMIN KOSRAT (SE) 2003-11-27 US disclosed
US-6579884-B1 Compounds ASTRAZENECA AB (SE) 2003-06-17 US disclosed
CN-1100056-C Compound for inhibition of gastric acid secretion ASTRA AB (SE) 2003-01-29 CN disclosed
EP-0971920-B1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-6265415-B1 ANTIULCER AGENT ASTRAZENECA AB (SE) 2001-07-24 US disclosed
EP-1105391-A2 NEW COMPOUNDS AstraZeneca AB (SE) 2001-06-13 EP disclosed
CN-1248257-A Compound for inhibition of gastric acid secretion ASTRA AB (SE) 2000-03-22 CN disclosed
WO-2000011000-A2 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-03-02 WO disclosed
EP-0971920-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION Astra Aktiebolag (SE) 2000-01-19 EP disclosed
WO-1998037080-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRA AKTIEBOLAG (SE) 1998-08-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030220364-A1 New compounds SLC10A2, GIPR, FABP2 TSHR 2682/4885RAPGEF4 1067/4885SCN4A 2992/4885
US-20210403406-A1 PROCESS FOR PREPARING 2,6-DIALKYLPHENYLACETIC ACIDS ADH1C, ADH1A, ADH5 TSHR 4521/4885RAPGEF4 1649/4885SCN4A 724/4885
US-11691938-B2 Process for preparing 2,6-dialkylphenylacetic acids ADH1C, ADH1A, ADH5 TSHR 4521/4885RAPGEF4 1649/4885SCN4A 724/4885
US-20240002344-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR HISTONE LYSINE DEMETHYLASE INHIBITION KDM5C, KDM5B, KDM5A TSHR 4662/4885RAPGEF4 2692/4885SCN4A 3520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.