SCHEMBL6445664

SCHEMBL6445664

N#CCCNC(=O)C(CNC(=O)c1ccccc1[N+](=O)[O-])c1ccc(O)cc1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
CTSD P07339 1/20 0.43
HTT P42858 3/20 0.41
HPGD P15428 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
TDP1 Q9NUW8 3/20 0.39
ALPL P05186 2/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
ALPI P09923 1/20 0.38
ALPG P10696 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6472461 0.93 CTSD (0.46) ALDH1A1CTSDHTTHPGDMEN1
SCHEMBL6445280 0.90 CTSK (0.51) ALDH1A1CTSDHTTHPGDMEN1
SCHEMBL6443947 0.87 CTSD (0.41) ALDH1A1CTSDHTTHPGDMEN1
SCHEMBL6825007 0.85 KDM4E (0.47) ALDH1A1HTTMEN1KMT2ALMNA
SCHEMBL6447527 0.84 LMNA (0.41) ALDH1A1HPGDMEN1KMT2ALMNA
SCHEMBL6445609 0.83 CTSK (0.52) ALDH1A1CTSDHTTHPGDMEN1
SCHEMBL6443745 0.82 CTSS (0.47) CTSSCTSKGAANPC1RAB9A
SCHEMBL6443305 0.80 CTSD (0.46) ALDH1A1CTSDHTTHPGDMEN1
SCHEMBL6021168 0.80 CTSL (0.54) ALDH1A1CTSDLMNACTSSCTSK
SCHEMBL6444783 0.79 ALDH1A1 (0.47) ALDH1A1CTSDHTTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed