SCHEMBL6466063

SCHEMBL6466063

NC(=O)CC(CCC(C(=O)c1nc2ccccc2o1)c1ccccc1)c1ccccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
POLB P06746 1/20 0.41
CTSS P25774 8/20 0.38
GART P22102 1/20 0.37
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.36
ALDH1A1 P00352 1/20 0.36
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36
DAGLA Q9Y4D2 1/20 0.36
XDH P47989 4/20 0.36
RAB9A P51151 1/20 0.35
GLO1 Q04760 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466913 0.88 FAAH (0.41) KDM4EPOLBCTSSGARTALDH1A1
SCHEMBL7048984 0.80 KDM4E (0.40) KDM4EPOLBCTSSGARTMAPT
SCHEMBL6464310 0.77 ALDH1A1 (0.41) KDM4EPOLBCTSSGARTALDH1A1
SCHEMBL6463422 0.76 FAAH (0.41) CTSSGARTMAPTHTTFAAH
SCHEMBL7181305 0.75 LMNA (0.42) CTSSMAPTCYP3A4CYP2C9
SCHEMBL6471951 0.74 XDH (0.43) KDM4ECTSSGARTFAAHCES1
SCHEMBL6465893 0.73 GART (0.43) KDM4ECTSSGARTFAAHCES1
SCHEMBL6461911 0.71 FAAH (0.42) CTSSGARTMAPTHTTFAAH
SCHEMBL11078276 0.70 DCAF1 (0.43) MAPTALDH1A1
SCHEMBL6465159 0.68 FAAH (0.44) CTSSGARTALDH1A1FAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed