SCHEMBL6499003

SCHEMBL6499003

CCCOc1ccc(C(=O)NCc2cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn2)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 2/20 0.37
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
P2RX7 Q99572 1/20 0.35
ACACB O00763 1/20 0.34
ALDH1A1 P00352 1/20 0.34
S1PR3 Q99500 3/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
ROCK2 O75116 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504861 0.92 HPGD (0.39) HPGDRAB9ANPC1TP53MAPT
Trifluoroacetic Acid SCHEMBL6498995 0.89 PPARG (0.39) HPGDRAB9ANPC1TP53MAPT
SCHEMBL6505057 0.89 HPGD (0.48) HPGDRAB9ANPC1P2RX7KMT2A
SCHEMBL6497497 0.87 S1PR3 (0.38) HPGDRAB9AP2RX7S1PR3MEN1
Trifluoroacetic Acid SCHEMBL6504858 0.81 HPGD (0.40) HPGDRAB9AP2RX7ALDH1A1PPARG
Trifluoroacetic Acid SCHEMBL6505054 0.77 HPGD (0.49) HPGDRAB9AP2RX7ALDH1A1PPARG
Trifluoroacetic Acid SCHEMBL6497487 0.76 S1PR3 (0.40) S1PR3PPARGPPARA
SCHEMBL6504395 0.76 PPARA (0.37) MAPTP2RX7PPARGPPARDPPARA
SCHEMBL6505593 0.76 ADORA2A (0.35) HPGDRAB9ANPC1ALDH1A1PPARD
SCHEMBL6494741 0.75 PPARA (0.39) MAPTPPARGPPARDPPARAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed