SCHEMBL6505057

SCHEMBL6505057

CC(C)OC(Cc1ccnc(CNC(=O)c2ccc(Cl)cc2Cl)c1)C(=O)OC(=O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.48
RAB9A P51151 1/20 0.40
NPC1 O15118 1/20 0.38
KLKB1 P03952 1/20 0.38
P2RX7 Q99572 4/20 0.37
POLB P06746 1/20 0.37
THRB P10828 1/20 0.37
RECQL P46063 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KMT2A Q03164 2/20 0.37
ATM Q13315 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
EPHX2 P34913 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SLC6A9 P48067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504861 0.92 HPGD (0.39) HPGDRAB9ANPC1KLKB1P2RX7
SCHEMBL6499003 0.89 HPGD (0.37) HPGDRAB9ANPC1P2RX7RECQL
Trifluoroacetic Acid SCHEMBL6505054 0.88 HPGD (0.49) HPGDRAB9AKLKB1P2RX7POLB
SCHEMBL6497497 0.87 S1PR3 (0.38) HPGDRAB9AP2RX7KMT2AEPHX2
SCHEMBL6495822 0.85 SHMT1 (0.39) HPGDKLKB1KMT2AEPHX2
SCHEMBL6504395 0.83 PPARA (0.37) KLKB1P2RX7GAA
SCHEMBL6498709 0.80 CDK2 (0.34) NPC1KLKB1P2RX7
Trifluoroacetic Acid SCHEMBL6504858 0.80 HPGD (0.40) HPGDRAB9AP2RX7
SCHEMBL6505593 0.80 ADORA2A (0.35) HPGDRAB9ANPC1POLBHTT
SCHEMBL6505045 0.78 SMN1; SMN2 (0.35) HPGDRAB9ANPC1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed