SCHEMBL6504861

SCHEMBL6504861

CC(C)Oc1ccc(C(=O)NCc2cc(CC(OC(C)C)C(=O)OC(=O)C(F)(F)F)ccn2)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.39
RAB9A P51151 2/20 0.39
P2RX7 Q99572 1/20 0.36
PTGDR Q13258 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KLKB1 P03952 2/20 0.34
NPC1 O15118 2/20 0.33
NR1H4 Q96RI1 2/20 0.33
EPHX2 P34913 1/20 0.33
NAMPT P43490 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
HDAC3 O15379 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499003 0.92 HPGD (0.37) HPGDRAB9AP2RX7ALDH1A1NPC1
SCHEMBL6505057 0.92 HPGD (0.48) HPGDRAB9AP2RX7KLKB1NPC1
SCHEMBL6497497 0.90 S1PR3 (0.38) HPGDRAB9AP2RX7EPHX2MEN1
Trifluoroacetic Acid SCHEMBL6504858 0.88 HPGD (0.40) HPGDRAB9AP2RX7PTGDRALDH1A1
Trifluoroacetic Acid SCHEMBL6498995 0.81 PPARG (0.39) HPGDRAB9AALDH1A1NPC1TP53
Trifluoroacetic Acid SCHEMBL6505054 0.80 HPGD (0.49) HPGDRAB9AP2RX7ALDH1A1KLKB1
Trifluoroacetic Acid SCHEMBL6497487 0.79 S1PR3 (0.40)
SCHEMBL6504395 0.78 PPARA (0.37) P2RX7KLKB1MAPTSMN1; SMN2
SCHEMBL6505593 0.78 ADORA2A (0.35) HPGDRAB9AALDH1A1NPC1POLB
SCHEMBL6494741 0.78 PPARA (0.39) MAPTMEN1KMT2APOLBHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed