SCHEMBL653241

SCHEMBL653241

Nc1ccccc1NC(=O)O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 16/20 0.68
HDAC1 Q13547 16/20 0.68
HDAC2 Q92769 16/20 0.68
MAPK1 P28482 1/20 0.68
NCOR2 Q9Y618 7/20 0.59
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
HDAC10 Q969S8 8/20 0.58
HDAC6 Q9UBN7 7/20 0.58
HDAC4 P56524 6/20 0.58
HDAC7 Q8WUI4 6/20 0.58
HDAC11 Q96DB2 6/20 0.58
HDAC8 Q9BY41 6/20 0.58
HDAC9 Q9UKV0 6/20 0.58
HDAC5 Q9UQL6 6/20 0.58
PTGS1 P23219 1/20 0.51
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250263 0.84 HDAC3 (0.64) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL31174164 0.84 HDAC3 (0.64) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL3071688 0.84 HDAC3 (0.64) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL9515806 0.84 NPC1 (0.67) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL17796923 0.84 HDAC3 (0.50) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL1226530 0.83 SMN1; SMN2 (0.54) HDAC3HDAC1HDAC2MAPK1NPC1
SCHEMBL29519193 0.83 SMN1; SMN2 (0.54) HDAC3HDAC1HDAC2MAPK1NPC1
SCHEMBL11048016 0.83 HDAC3 (0.63) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL407834 0.81 HDAC1 (1.00) HDAC3HDAC1HDAC2MAPK1NCOR2
SCHEMBL30363156 0.81 HDAC1 (1.00) HDAC3HDAC1HDAC2MAPK1NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293718-B1 SUBSTITUTED AMINOPHENYL CARBAMATE BAYER AG (DE) 1993-02-03 EP claimed
EP-0293718-A2 Substituted aminophenyl carbamate BAYER AG (DE) 1988-12-07 EP claimed
WO-2024148329-A1 LIPID CONJUGATES FOR THE DELIVERY OF THERAPEUTIC AGENTS TO ADIPOSE TISSUE Arrowhead Pharmaceuticals, Inc. (US) 2024-07-11 WO disclosed
WO-2023242070-A9 ANTIMICROBIAL COMPOUNDS AKTHELIA PHARMACEUTICALS (IS) 2024-06-20 WO disclosed
WO-2024123929-A1 DEVELOPMENT OF POTENT DUAL HDAC/BRD4 INHIBITORS BIOVENTURES, LLC (US) 2024-06-13 WO disclosed
EP-4093730-B1 HDAC DEGRADER UNIV LEICESTER (GB) 2024-05-08 EP disclosed
WO-2023242070-A1 ANTIMICROBIAL COMPOUNDS AKTHELIA PHARMACEUTICALS (IS) 2023-12-21 WO disclosed
US-11772085-B2 Far superior oxidation catalysts based on macrocyclic compounds CARNEGIE MELLON UNIVERSITY (US) 2023-10-03 US disclosed
US-11655260-B2 Heterocyclic compounds as arginase inhibitors GUANGDONG NEWOPP BIOPHARMACEUTICALS CO., LTD. (CN) 2023-05-23 US disclosed
US-20230120211-A1 HDAC Degrader UNIVERSITY OF LEICESTER (GB) 2023-04-20 US disclosed
US-20230113588-A1 METABOTROPIC GLUTAMATE RECEPTOR NEGATIVE ALLOSTERIC MODULATORS (NAMS) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute 2023-04-13 US disclosed
US-6090525-A PHOTOSENSITIVE POLYIMIDE COATING AGENT COMPOSITION WITH BOTH GOOD VISCOSITY STABILITY AT ROOM TEMPERATURE WITH LAPSE OF TIME AND GOOD PHOTOSENSITIVE PERFORMANCE TORAY INDUSTRIES, INC. (JP) 2000-07-18 US disclosed
EP-0878740-A1 Radiation sensitive polymer composition TORAY INDUSTRIES, INC. (JP) 1998-11-18 EP disclosed
EP-0293718-B1 SUBSTITUTED AMINOPHENYL CARBAMATE BAYER AG (DE) 1993-02-03 EP disclosed
EP-0293718-B1 SUBSTITUTED AMINOPHENYL CARBAMATE BAYER AG (DE) 1993-02-03 EP disclosed
EP-0293718-A2 Substituted aminophenyl carbamate BAYER AG (DE) 1988-12-07 EP disclosed
EP-0293718-A2 Substituted aminophenyl carbamate BAYER AG (DE) 1988-12-07 EP disclosed
EP-0293718-A2 Substituted aminophenyl carbamate BAYER AG (DE) 1988-12-07 EP disclosed
US-4241218-A TOXIC AGENTS FOR CHEMICAL WARFARE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1980-12-23 US disclosed
US-3979202-A Meta-bifunctional benzenes and herbicidal compositions MONSANTO COMPANY (US) 1976-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11655260-B2 Heterocyclic compounds as arginase inhibitors ARG1, ARG2, PRMT1 HDAC3 195/4885HDAC1 62/4885HDAC2 104/4885
US-11772085-B2 Far superior oxidation catalysts based on macrocyclic compounds SOD1, ME3, ME2 HDAC3 1378/4885HDAC1 800/4885HDAC2 1796/4885
US-20230120211-A1 HDAC Degrader HDAC1, HDAC11, HDAC3 HDAC3 3/4885HDAC1 1/4885HDAC2 4/4885
US-20230113588-A1 METABOTROPIC GLUTAMATE RECEPTOR NEGATIVE ALLOSTERIC MODULATORS (NAMS) AND USES THEREOF GRM3, GRM2, GRM1 HDAC3 239/4885HDAC1 657/4885HDAC2 571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.