Decitabine

Decitabine

SCHEMBL661233

Nc1ncn([C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DNMT1DNMT3A

The experimentally established mechanism targets of Decitabine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 known ✓ P26358 5/20 1.00
ADRB1 P08588 1/20 1.00
LMNA P02545 3/20 0.62
TP53 P04637 2/20 0.62
HTT P42858 2/20 0.62
GMNN O75496 1/20 0.62
ALDH1A1 P00352 1/20 0.62
NFKB1 P19838 1/20 0.62
THPO P40225 1/20 0.62
MTOR P42345 1/20 0.62
RAB9A P51151 1/20 0.62
BLM P54132 1/20 0.62
HBB P68871 1/20 0.62
PMP22 Q01453 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.57
PNP P00491 1/20 0.57
PDE4D Q08499 1/20 0.57
PDE3A Q14432 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57
PIM1 P11309 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Decitabine SCHEMBL10030513 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL9999636 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL172264 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL1651086 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL4006 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL117721 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL12800474 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL20651628 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL20769771 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT
Decitabine SCHEMBL18402620 1.00 DNMT1 (1.00) DNMT1ADRB1LMNATP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 230 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050118600-A1 Method for selecting drug sensitivity-determining factors and method for predicting drug sensitivity using the selected factors F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 US claimed
US-20030138864-A1 Method for identifying an enzyme to design anti-cancer compounds CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-07-24 US claimed
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-03-17 US disclosed
US-12441708-B2 Cereblon ligands and bifunctional compounds comprising the same ARVINAS OPERATIONS, INC. (US) 2025-10-14 US disclosed
US-20250313547-A1 CEREBLON LIGANDS AND BIFUNCTIONAL COMPOUNDS COMPRISING THE SAME ARVINAS OPERATIONS INC (US) 2025-10-09 US disclosed
US-12251402-B2 Mesenchymal stem cells with enhanced immunosuppressive capability ESCAPE THERAPEUTICS, INC. (US) 2025-03-18 US disclosed
US-20250000887-A1 COMPOSITIONS COMPRISING 2'-DEOXYCYTIDINE ANALOGS AND USE THEREOF FOR THE TREATMENT OF SICKLE CELL DISEASE, THALASSEMIA, AND CANCERS AKIRABIO, INC. (US) 2025-01-02 US disclosed
US-20240301054-A1 TIM-3 INHIBITORS AND USES THEREOF NOVARTIS AG (CH) 2024-09-12 US disclosed
US-20240301053-A1 COMBINATION THERAPIES WITH VENETOCLAX AND TIM-3 INHIBITORS NOVARTIS AG (CH) 2024-09-12 US disclosed
US-12023385-B2 Tunable endogenous protein degradation with heterobifunctional compounds DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-07-02 US disclosed
US-12011432-B2 Method of modulating ribonucleotide reductase CASE WESTERN RESERVE UNIVERSITY (US) 2024-06-18 US disclosed
WO-2008101448-A2 METHOD OF MANUFACTURING 1-(2-DEOXY-ALPHA-D-ERYTHRO-PENTOFURANOSYL)-5-AZACYTOSINE USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2008-08-28 WO disclosed
WO-2008101448-A2 METHOD OF MANUFACTURING 1-(2-DEOXY-ALPHA-D-ERYTHRO-PENTOFURANOSYL)-5-AZACYTOSINE USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2008-08-28 WO disclosed
US-20080182806-A1 USE OF ACETYLATED OR ESTERIFICATED AZACYTIDINE, DECITABINE, OR OTHER NUCLEOSIDE ANALOGS AS ORAL AGENTS FOR THE TREATMENT OF TUMORS OR OTHER DYSPLASTIC SYNDROMES SENSITIVE TO HYPOMETHYLATING AGENTS NEVADA CANCER INSTITUTE (US) 2008-07-31 US disclosed
WO-2008092127-A1 USE OF ACETYLATED OR ESTERIFICATED AZACYTIDINE, DECITABINE, OR OTHER NUCLEOSIDE ANALOGS AS ORAL AGENTS FOR THE TREATMENT OF TUMORS OR OTHER DYSPLASTIC SYNDROMES SENSITIVE TO HYPOMETHYLATING AGENTS NEVADA CANCER INSTITUTE (US) 2008-07-31 WO disclosed
WO-2008083634-A1 1-(2-DEOXY-ALPHA-D-ERYTHRO-PENTOFURANOSYL)-5-AZACYTOSINE FOR USE AS DRUG USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2008-07-17 WO disclosed
WO-2008083634-A1 1-(2-DEOXY-ALPHA-D-ERYTHRO-PENTOFURANOSYL)-5-AZACYTOSINE FOR USE AS DRUG USTAV ORGANICKE CHEMIE A BIOCHEMIE AV CR, V.V.I. (CZ) 2008-07-17 WO disclosed
US-20070117776-A1 Low Dose Therapy Of DNA Methylation Inhibitors SUPERGEN, INC. 2007-05-24 US disclosed
US-20050118600-A1 Method for selecting drug sensitivity-determining factors and method for predicting drug sensitivity using the selected factors F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 US disclosed
US-20030138864-A1 Method for identifying an enzyme to design anti-cancer compounds CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-07-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030138864-A1 Method for identifying an enzyme to design anti-cancer compounds RNASE1, GUSB, DPEP1 DNMT1 2168/4885ADRB1 4416/4885LMNA 4056/4885
US-20250313547-A1 CEREBLON LIGANDS AND BIFUNCTIONAL COMPOUNDS COMPRISING THE SAME CRBN, CBL, MDM2 DNMT1 2907/4885ADRB1 4482/4885LMNA 3085/4885
US-20240301054-A1 TIM-3 INHIBITORS AND USES THEREOF HAVCR2, CD58, LGALS3 DNMT1 2930/4885ADRB1 3784/4885LMNA 2642/4885
US-12023385-B2 Tunable endogenous protein degradation with heterobifunctional compounds DBN1, MYCBP, PSMG3 DNMT1 3525/4885ADRB1 4535/4885LMNA 2907/4885
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use MDM2, UBR4, UBE3A DNMT1 1975/4885ADRB1 4096/4885LMNA 2705/4885
US-20250000887-A1 COMPOSITIONS COMPRISING 2'-DEOXYCYTIDINE ANALOGS AND USE THEREOF FOR THE TREATMENT OF SICKLE CELL DISEASE, THALASSEMIA, AND CANCERS TYMP, HBZ, HBB DNMT1 111/4885ADRB1 2700/4885LMNA 835/4885
US-12251402-B2 Mesenchymal stem cells with enhanced immunosuppressive capability HLA-C, HLA-B, HLA-DRB1 DNMT1 7/4885ADRB1 2511/4885LMNA 3899/4885
US-20240301053-A1 COMBINATION THERAPIES WITH VENETOCLAX AND TIM-3 INHIBITORS HAVCR2, BCL3, BIRC3 DNMT1 2240/4885ADRB1 3969/4885LMNA 2056/4885
US-12011432-B2 Method of modulating ribonucleotide reductase RRM2, RRM2B, RRM1 DNMT1 513/4885ADRB1 2260/4885LMNA 3520/4885
US-12441708-B2 Cereblon ligands and bifunctional compounds comprising the same CRBN, CBL, MDM2 DNMT1 2907/4885ADRB1 4482/4885LMNA 3085/4885
US-20080182806-A1 USE OF ACETYLATED OR ESTERIFICATED AZACYTIDINE, DECITABINE, OR OTHER NUCLEOSIDE ANALOGS AS ORAL AGENTS FOR THE TREATMENT OF TUMORS OR OTHER DYSPLASTIC SYNDROMES SENSITIVE TO HYPOMETHYLATING AGENTS DCTD, DNMT3A, HDAC5 DNMT1 5/4885ADRB1 4614/4885LMNA 939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.