SCHEMBL6633602

SCHEMBL6633602

CC(C)CC(=O)N(C(=O)N(Cc1ccccc1)[C@@H]1CCCNCC1=O)S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.40
SLC6A4 P31645 12/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KCNH2 Q12809 7/20 0.37
SLC6A3 Q01959 7/20 0.37
CNR2 P34972 1/20 0.35
MCL1 Q07820 4/20 0.35
STAT3 P40763 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
PKM P14618 1/20 0.35
BCL2L1 Q07817 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430902 0.73 ALDH1A1 (0.38) SLC6A2SLC6A4SMN1; SMN2ALDH1A1GAA
SCHEMBL4767101 0.71 CTSD (0.37) SLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL6770905 0.70 GHSR (0.38) SLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL6588875 0.67 CTSK (0.39)
SCHEMBL4936544 0.67 GHSR (0.37) SLC6A2SLC6A4SLC6A3
SCHEMBL4766714 0.67 GHSR (0.37) SLC6A2SLC6A4SLC6A3
SCHEMBL7570056 0.67 OPRM1 (0.47) SLC6A2SLC6A4SMN1; SMN2ALDH1A1GAA
SCHEMBL7562358 0.67 ACKR3 (0.45) SLC6A2SLC6A4SMN1; SMN2ALDH1A1GAA
SCHEMBL7538627 0.66 ALDH1A1 (0.39) SMN1; SMN2STAT3ALDH1A1LMNAGAA
SCHEMBL7564716 0.66 PSEN1 (0.34) SLC6A2SLC6A4KCNH2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed