SCHEMBL7562358

SCHEMBL7562358

C[C@@H](CCNC(=O)c1cc2ccccc2o1)CC(=O)N(Cc1ccccc1)C1CCCNCC1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.45
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
ALDH1A1 P00352 6/20 0.40
HPGD P15428 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TP53 P04637 2/20 0.40
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 2/20 0.39
DRD3 P35462 2/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
HDAC3 O15379 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570056 0.83 OPRM1 (0.47) OPRM1OPRK1TMEM97SIGMAR1SLC6A2
SCHEMBL4767101 0.78 CTSD (0.37) OPRM1SLC6A2SLC6A4MEN1KMT2A
SCHEMBL7426386 0.71 RAB9A (0.45) HPGDSMN1; SMN2TP53RAB9ANPC1
SCHEMBL7430902 0.70 ALDH1A1 (0.38) SLC6A2SLC6A4ALDH1A1HPGDSMN1; SMN2
SCHEMBL4763259 0.69 CTSD (0.44) SLC6A2SLC6A4ALDH1A1MEN1KMT2A
SCHEMBL6404263 0.69 CTSK (0.50)
SCHEMBL6590467 0.69 CTSK (0.42) SMN1; SMN2TP53RAB9ANPC1MEN1
SCHEMBL6770905 0.69 GHSR (0.38) SLC6A2SLC6A4
SCHEMBL4766714 0.67 GHSR (0.37) SLC6A2SLC6A4HPGD
SCHEMBL4936544 0.67 GHSR (0.37) SLC6A2SLC6A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed