SCHEMBL6835178

SCHEMBL6835178

CC(=C(C#N)C#N)c1ccccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.62
GABRG2 P18507 4/20 0.62
GABRB3 P28472 4/20 0.62
GABRB2 P47870 3/20 0.62
GABRB1 P18505 1/20 0.62
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TRPA1 O75762 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 2/20 0.39
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38
MAPK1 P28482 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320966 0.78 KMT2A (0.47) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL21056095 0.77 GABRA1 (1.00) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL29061079 0.76 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL9824671 0.74 CES2 (0.50) CES2CES1ALDH1A1POLBKMT2A
SCHEMBL8532480 0.73 POLB (0.41) CES2CES1ALDH1A1TRPA1NPSR1
SCHEMBL28260941 0.73 NR4A1 (0.46) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL7308873 0.73 CTSD (0.43) GABRA1GABRG2GABRB3GABRB2GABRB1
SCHEMBL9487828 0.72 CES2 (0.48) CES2CES1ALDH1A1POLBKMT2A
SCHEMBL25680264 0.72 CES2 (0.48) CES2CES1ALDH1A1POLBKMT2A
SCHEMBL25680262 0.72 CES2 (0.48) CES2CES1ALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116496191-A Preparation method of polysubstituted alkenyl thioether compound 浙江大学 2023-07-28 CN disclosed
CN-108947890-B Method for preparing disubstituted 4-aminocarbazole compound 台州学院 2020-08-04 CN disclosed
US-9951020-B2 Methods of making 2-halonicotinonitriles VIRGINIA COMMONWEALTH UNIVERSITY (US) 2018-04-24 US disclosed
US-9951020-B2 Methods of making 2-halonicotinonitriles VIRGINIA COMMONWEALTH UNIVERSITY (US) 2018-04-24 US disclosed
US-20160221951-A1 METHODS OF MAKING 2-HALONICOTINONITRILES VIRGINIA COMMONWEALTH UNIVERSITY 2016-08-04 US disclosed
US-20160221951-A1 METHODS OF MAKING 2-HALONICOTINONITRILES VIRGINIA COMMONWEALTH UNIVERSITY 2016-08-04 US disclosed
WO-2015031718-A1 METHODS OF MAKING 2-HALONICOTINONITRILES MCQUADE D TYLER (US) 2015-03-05 WO disclosed
CN-1523958-A Pesticide compositions comprising malononitrile compounds ס�ѻ�ѧ��ҵ��ʽ���� 2004-08-25 CN disclosed
US-20040142821-A1 Pesticide composition comprising malononitrile compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221951-A1 METHODS OF MAKING 2-HALONICOTINONITRILES NISCH, HCN2, HCN1 GABRA1 4531/4885GABRG2 4492/4885GABRB3 4288/4885
US-20040142821-A1 Pesticide composition comprising malononitrile compounds CBR1, CBR3, ME1 GABRA1 3081/4885GABRG2 4022/4885GABRB3 3691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.