SCHEMBL6853374

SCHEMBL6853374

c1ccc(-c2nc3ccccc3cc2CN2CCN(C3CCCCC3)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 7/20 0.50
KCNH2 Q12809 1/20 0.50
TACR2 P21452 6/20 0.49
OPRM1 P35372 3/20 0.49
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TP53 P04637 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
SIGMAR1 Q99720 3/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TRPV4 Q9HBA0 2/20 0.42
ABCB1 P08183 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6851652 0.84 TACR3 (0.50) TACR3KCNH2TACR2OPRM1ALDH1A1
SCHEMBL6854970 0.81 KMT2A (0.50) KCNH2DRD4DRD3ALDH1A1KDM4E
SCHEMBL5945358 0.81 SLC2A1 (0.46) TACR3TACR2OPRM1
SCHEMBL6853013 0.80 HRH3 (0.48) ALDH1A1KDM4EHRH3KMT2A
SCHEMBL6853531 0.80 DRD2 (0.50) DRD4DRD3ALDH1A1KDM4EMEN1
SCHEMBL6848935 0.77 SLC2A1 (0.44) TACR3KCNH2TACR2OPRM1ALDH1A1
SCHEMBL6853077 0.77 HTR2B (0.49) DRD4DRD3ALDH1A1KDM4ESIGMAR1
SCHEMBL5908682 0.77 FAAH (0.42) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL6848678 0.77 TACR2 (0.53) TACR3KCNH2TACR2OPRM1HRH3
SCHEMBL5442168 0.77 PDE10A (0.43) ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US disclosed