SCHEMBL692620

SCHEMBL692620

O=C(O)c1[c]c(O)cc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
HPGD P15428 4/20 0.50
ALDH1A1 P00352 3/20 0.50
HSD17B10 Q99714 3/20 0.50
KDM4E B2RXH2 2/20 0.50
CYP1A2 P05177 1/20 0.50
GLA P06280 1/20 0.50
CYP2C19 P33261 1/20 0.50
TRPM4 Q8TD43 1/20 0.44
GPR35 Q9HC97 2/20 0.44
POLB P06746 1/20 0.44
CDC25B P30305 2/20 0.42
LDHA P00338 1/20 0.42
CYP2D6 P10635 1/20 0.41
NR4A1 P22736 1/20 0.41
NR4A2 P43354 1/20 0.41
NR4A3 Q92570 1/20 0.41
GRIN2D O15399 1/20 0.40
GRIN2A Q12879 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5411002 0.84 KDM4E (0.43) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL5032934 0.76 TRPM4 (0.48) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL29019737 0.71 TRPM4 (0.43) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL7628474 0.70 ERN1 (0.42) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL9770151 0.70 MEN1 (0.50) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL770722 0.69 CYP1A2 (0.70) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL2517773 0.69 NR4A1 (0.48) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL6631799 0.69 CYP2D6 (0.47) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL6461 0.68 ACMSD (0.39) MEN1KMT2AHPGDALDH1A1HSD17B10
SCHEMBL245378 0.68 CYP1A2 (0.62) MEN1KMT2AHPGDALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130122073-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANANCE OF CONTACT LENSES AND MEDICAL MATERIALS UNIWERSYTET JAGIELLONSKI (PL) 2013-05-16 US claimed
EP-2563148-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANCE OF CONTACT LENSES AND MEDICAL MATERIALS Uniwersytet Jagiellonski (PL) 2013-03-06 EP claimed
US-20120071428-A1 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE JAGIELLONIAN UNIVERSITY (PL) 2012-03-22 US claimed
EP-2421644-A2 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE Uniwersytet Jagiello Ski (PL) 2012-02-29 EP claimed
WO-2011136672-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANCE OF CONTACT LENSES AND MEDICAL MATERIALS Uniwersytet Jagielloński (PL) 2011-11-03 WO claimed
WO-2010098687-A2 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE Uniwersytet Jagielloński (PL) 2010-09-02 WO claimed
EP-2421644-B1 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE UNIV JAGIELLONSKI (PL) 2019-07-17 EP disclosed
EP-3089818-B1 A VISIBLE-LIGHT-ACTIVATED MULTILAYERED PHOTOCATALYST AND THE METHOD OF ITS PREPARATION UNIV JAGIELLONSKI (PL) 2018-05-23 EP disclosed
US-20170001183-A1 Visible-Light-Activated Multilayered Photocatalyst And The Method Of Its Preparation UNIWERSYTET JAGIELLONSKI (PL) 2017-01-05 US disclosed
EP-3089818-A2 A VISIBLE-LIGHT-ACTIVATED MULTILAYERED PHOTOCATALYST AND THE METHOD OF ITS PREPARATION Uniwersytet Jagiellonski (PL) 2016-11-09 EP disclosed
EP-2563148-B1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANCE OF CONTACT LENSES AND MEDICAL MATERIALS UNIV JAGIELLONSKI (PL) 2016-08-24 EP disclosed
US-9040489-B2 Nanocrystalline photocatalytic colloid, a method of producing it and its use JAGIELLONIAN UNIVERSITY (PL) 2015-05-26 US disclosed
US-20130122073-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANANCE OF CONTACT LENSES AND MEDICAL MATERIALS UNIWERSYTET JAGIELLONSKI (PL) 2013-05-16 US disclosed
EP-2563148-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANCE OF CONTACT LENSES AND MEDICAL MATERIALS Uniwersytet Jagiellonski (PL) 2013-03-06 EP disclosed
US-20120071428-A1 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE JAGIELLONIAN UNIVERSITY (PL) 2012-03-22 US disclosed
EP-2421644-A2 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE Uniwersytet Jagiello Ski (PL) 2012-02-29 EP disclosed
WO-2011136672-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANCE OF CONTACT LENSES AND MEDICAL MATERIALS Uniwersytet Jagielloński (PL) 2011-11-03 WO disclosed
US-20100323202-A1 USE OF CARBOXYLIC ACID HYDRAZIDE FOR DE-BONDING POLYURETHANE ADHESIVES SIKA TECHNOLOGY AG (CH) 2010-12-23 US disclosed
US-20100273924-A1 CURABLE COMPOSITIONS HAVING LESS VOLATILIZATION SIKA TECHNOLOGY AG (CH) 2010-10-28 US disclosed
WO-2010098687-A2 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE Uniwersytet Jagielloński (PL) 2010-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120071428-A1 NANOCRYSTALLINE PHOTOCATALYTIC COLLOID, A METHOD OF PRODUCING IT AND ITS USE UROD, CRYZ, CRYAB MEN1 1615/4885KMT2A 3369/4885HPGD 3914/4885
US-20130122073-A1 COMPOSITION IN THE FORM OF LIQUID FOR MAINTENANANCE OF CONTACT LENSES AND MEDICAL MATERIALS MLEC, CRYZ, LAGE3 MEN1 262/4885KMT2A 1127/4885HPGD 1510/4885
US-20100273924-A1 CURABLE COMPOSITIONS HAVING LESS VOLATILIZATION CA4, CTH, CA6 MEN1 1018/4885KMT2A 294/4885HPGD 2018/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.