SCHEMBL6959326

SCHEMBL6959326

N#Cc1cccc(CNc2cnn(-c3ccccc3)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 3/20 0.51
GRM5 P41594 1/20 0.47
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
LRRK2 Q5S007 1/20 0.45
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
TSHR P16473 1/20 0.45
NTRK1 P04629 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44
CLK4 Q9HAZ1 2/20 0.44
NOS1 P29475 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969995 0.78 ACP1 (0.45) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6959537 0.77 VNN1 (0.48) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6959349 0.76 VNN1 (0.47) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6960930 0.76 VNN1 (0.47) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6691560 0.76 NOS1 (0.58) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1680823 0.74 LMNA (0.57) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2214866 0.72 GAA (0.53) GRM5TSHR
SCHEMBL6972135 0.72 MEN1 (0.47) VNN1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6966037 0.72 ALKBH1 (0.43) VNN1GRM5ALDH1A1HSD17B10ALKBH1
SCHEMBL19902102 0.71 GRM5 (0.70) GRM5GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed