SCHEMBL6972036

SCHEMBL6972036

CN(Cc1ccc(Cc2c[nH]cn2)cc1)C(=O)Cc1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
HTT P42858 1/20 0.50
RAB9A P51151 1/20 0.50
CNR2 P34972 4/20 0.40
ERCC1 P07992 1/20 0.40
ERCC4 Q92889 1/20 0.40
ROCK2 O75116 1/20 0.39
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CNR1 P21554 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
THRB P10828 1/20 0.37
AOC3 Q16853 1/20 0.36
P2RX7 Q99572 1/20 0.36
CXCR3 P49682 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9080507 0.90 AOC3 (0.45) ALDH1A1HTTRAB9AERCC1ERCC4
SCHEMBL6961731 0.89 ALDH1A1 (0.49) ALDH1A1HTTRAB9ACNR2ERCC1
SCHEMBL6966973 0.89 ROCK2 (0.50) ALDH1A1RAB9AROCK2NPC1SMN1; SMN2
SCHEMBL6966618 0.89 ALDH1A1 (0.47) ALDH1A1HTTRAB9ANPC1SMN1; SMN2
SCHEMBL6974366 0.88 LTB4R (0.45) ALDH1A1HTTRAB9AAOC3CXCR3
SCHEMBL6969265 0.83 ALDH1A1 (0.41) ALDH1A1HTTRAB9ANPC1SMN1; SMN2
SCHEMBL9079317 0.83 CCR5 (0.37) CNR2
SCHEMBL6970199 0.81 RAB9A (0.40) ALDH1A1HTTRAB9ACNR2NPC1
SCHEMBL9024045 0.81 AOC3 (0.41) ALDH1A1HTTRAB9ANPC1SMN1; SMN2
SCHEMBL6973527 0.80 LTB4R (0.46) ALDH1A1HTTRAB9AAOC3CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729459-B1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORP (US) 2003-03-12 EP disclosed
US-5578616-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, TREATMENT FOR GASTROINTESTINAL AND CARDIOVASCULAR DISORDERS SCHERING CORPORATION (US) 1996-11-26 US disclosed
EP-0729459-A1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 1996-09-04 EP disclosed
WO-1995014007-A1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 1995-05-26 WO disclosed