SCHEMBL6976687

SCHEMBL6976687

CC1=C(C)C2=C(N)C(C)(CN3CCC(c4cn(-c5ccccc5)c5ccccc45)CC3)CC2=C(C)O1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.39
HTR6 P50406 4/20 0.34
DRD2 P14416 1/20 0.32
HRH2 P25021 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981567 0.81 DRD2 (0.40) DRD2
Hydrochloric Acid SCHEMBL6985853 0.80 DRD2 (0.40) DRD2
Hydrochloric Acid SCHEMBL6984760 0.80 DRD2 (0.40) DRD2
SCHEMBL6985176 0.79 HTR6 (0.39) KCNH2HTR6DRD2
Hydrochloric Acid SCHEMBL6986246 0.79 ADRA1D (0.46)
SCHEMBL6983492 0.77 CHRNA7 (0.40) KCNH2DRD2
SCHEMBL6979708 0.76 PRMT6 (0.43) KCNH2
SCHEMBL6981079 0.73 HRH3 (0.40)
Hydrochloric Acid SCHEMBL6979051 0.72 LMNA (0.41) DRD2
SCHEMBL6976685 0.72 KCNH2 (0.38) KCNH2HTR6HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed