SCHEMBL6978202

SCHEMBL6978202

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)C4CC4)c32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
GAA P10253 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
DPP8 Q6V1X1 1/20 0.37
DPP9 Q86TI2 1/20 0.37
FPR1 P21462 2/20 0.36
FPR2 P25090 2/20 0.36
ATM Q13315 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NR3C1 P04150 1/20 0.35
AR P10275 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981035 0.96 DPP8 (0.36) ALDH1A1GAASMN1; SMN2DPP8DPP9
SCHEMBL6978509 0.86 PTGER4 (0.40) ALDH1A1GAASMN1; SMN2DPP8DPP9
SCHEMBL6985322 0.86 GAA (0.41) ALDH1A1GAAFPR1FPR2HDAC1
SCHEMBL6985566 0.86 PARP14 (0.40) ALDH1A1SMN1; SMN2DPP8DPP9FPR1
SCHEMBL6982945 0.85 NR3C1 (0.36) ALDH1A1GAASMN1; SMN2DPP8DPP9
SCHEMBL6986437 0.84 PTGER4 (0.41) ALDH1A1SMN1; SMN2DPP8DPP9FPR1
SCHEMBL6984039 0.84 TP53 (0.45) ALDH1A1GAANR3C1ARMAPT
SCHEMBL6977498 0.84 CCKBR (0.44) ALDH1A1GAAHDAC1HDAC8HDAC6
SCHEMBL6984759 0.83 LMNA (0.47) ALDH1A1GAASMN1; SMN2KMT2AMEN1
SCHEMBL6982761 0.83 HDAC1 (0.35) ALDH1A1GAASMN1; SMN2DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed