SCHEMBL6981035

SCHEMBL6981035

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)C4CCCCC4)c32)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
ALDH1A1 P00352 4/20 0.35
MAPT P10636 1/20 0.35
FPR1 P21462 2/20 0.35
FPR2 P25090 2/20 0.35
ATM Q13315 1/20 0.35
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NR3C1 P04150 2/20 0.34
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978202 0.96 ALDH1A1 (0.37) DPP8DPP9ALDH1A1MAPTFPR1
SCHEMBL6985322 0.84 GAA (0.41) ALDH1A1MAPTFPR1FPR2GAA
SCHEMBL6978509 0.84 PTGER4 (0.40) DPP8DPP9ALDH1A1MAPTFPR1
SCHEMBL6985566 0.84 PARP14 (0.40) DPP8DPP9ALDH1A1MAPTFPR1
SCHEMBL6982945 0.83 NR3C1 (0.36) DPP8DPP9ALDH1A1MAPTFPR1
SCHEMBL6986437 0.82 PTGER4 (0.41) DPP8DPP9ALDH1A1MAPTFPR1
SCHEMBL6984039 0.82 TP53 (0.45) ALDH1A1MAPTGAANR3C1AR
SCHEMBL6977498 0.82 CCKBR (0.44) ALDH1A1MAPTGAAHDAC1HDAC8
SCHEMBL6985749 0.82 ALDH1A1 (0.48) ALDH1A1MAPTGAAMEN1KMT2A
SCHEMBL6982764 0.82 FPR1 (0.43) ALDH1A1MAPTFPR1FPR2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed