SCHEMBL6988039

SCHEMBL6988039

CC(C)C[C@@H](C(=O)NN)[C@H](C(=O)NO)C(CNC(=O)c1ccccc1)(CC(C)C)C(=O)Cn1ccnc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 4/20 0.36
TBXAS1 P24557 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
ADAM17 P78536 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34
CYP19A1 P11511 1/20 0.34
HMOX2 P30519 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
HRH4 Q9H3N8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987467 0.94 CYP26A1 (0.36) CYP26A1TBXAS1CYP1A2CYP3A4CYP2D6
SCHEMBL6981901 0.90 HRH4 (0.39) CYP26A1TBXAS1CYP19A1FNTAFNTB
SCHEMBL6986413 0.90 CYP26A1 (0.37) CYP26A1TBXAS1CYP1A2CYP3A4CYP2D6
SCHEMBL7808546 0.89 CTSS (0.36) MMP2MMP9MMP8ADAM17HMOX2
SCHEMBL6987186 0.86 TBXAS1 (0.37) TBXAS1MMP2MMP9MMP8ADAM17
SCHEMBL7818934 0.83 CTSS (0.37) CYP3A4CYP2D6HMOX2FNTAFNTB
SCHEMBL7816193 0.80 CTSS (0.35) MMP8HMOX2
SCHEMBL6982695 0.79 CTSS (0.33) MMP8HMOX2
SCHEMBL6985861 0.79 HMOX2 (0.35) TBXAS1MMP2MMP9MMP8ADAM17
SCHEMBL7816001 0.79 CTSK (0.41) CYP19A1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed