SCHEMBL7159598

SCHEMBL7159598

COc1ccc(-c2nc(CO)c[nH]2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.45
PTGS2 P35354 5/20 0.39
PTGS1 P23219 2/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CHEK2 O96017 2/20 0.38
GRIN2B Q13224 1/20 0.38
S1PR4 O95977 1/20 0.38
KDM4E B2RXH2 2/20 0.38
PRKAB2 O43741 2/20 0.38
PRKAG1 P54619 2/20 0.38
PRKAA2 P54646 2/20 0.38
PRKAA1 Q13131 2/20 0.38
PRKAG3 Q9UGI9 2/20 0.38
PRKAG2 Q9UGJ0 2/20 0.38
PRKAB1 Q9Y478 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MPI P34949 1/20 0.38
GFER P55789 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7161302 0.89 KMO (0.43) KMOKDM4EPRKAB2PRKAG1PRKAA2
SCHEMBL7159559 0.83 ALDH1A1 (0.47) PTGS2PTGS1KDM4EALDH1A1GAA
SCHEMBL10556563 0.77 PTGS2 (0.47) KMOPTGS2PTGS1ADORA2AADORA1
SCHEMBL7422530 0.76 PDE4A (0.53)
SCHEMBL10556612 0.76 KDM4E (0.46) KDM4EALDH1A1GAAMPIGFER
SCHEMBL5801973 0.75 HTR7 (0.44) PDGFRBPDGFRA
SCHEMBL10355347 0.74 DCUN1D1 (0.49) ADORA2AADORA1KDM4ETDP1
SCHEMBL6859787 0.74 AMY1A (0.49) KDM4EALDH1A1GAAGFERTDP1
SCHEMBL23778736 0.74 NOTUM (0.45) PTGS2KDM4EALDH1A1GFER
SCHEMBL29008478 0.73 KDM4E (0.48) KDM4EALDH1A1GAAMPIGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358165-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-05 EP disclosed
WO-2002060877-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-08 WO disclosed