SCHEMBL718238

SCHEMBL718238

CCCCCCCCC=CCCCCCCCC(=O)NC(CC)N1CCN(C(CC)NC(=O)CCCCCCCC=CCCCCCCCC)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.57
ASAH2 Q9NR71 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SLC6A5 Q9Y345 1/20 0.53
DEGS1 O15121 1/20 0.53
ALDH1A1 P00352 1/20 0.52
CETP P11597 1/20 0.52
TP53 P04637 1/20 0.52
CNR2 P34972 3/20 0.51
TRPV1 Q8NER1 3/20 0.51
CNR1 P21554 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29245563 1.00 FAAH (0.57) FAAHASAH2SMN1; SMN2SLC6A5DEGS1
SCHEMBL10723388 0.91 FAAH (0.58) FAAHALDH1A1CNR2TRPV1CNR1
SCHEMBL5673619 0.82 FAAH (0.64) FAAHASAH2SLC6A5DEGS1ALDH1A1
SCHEMBL5673658 0.82 FAAH (0.64) FAAHASAH2SLC6A5DEGS1ALDH1A1
SCHEMBL8435127 0.81 ALDH1A1 (0.54) FAAHSMN1; SMN2ALDH1A1TP53CNR1
SCHEMBL1514267 0.81 ALDH1A1 (0.54) FAAHSMN1; SMN2ALDH1A1TP53CNR1
SCHEMBL8435136 0.81 ALDH1A1 (0.54) FAAHSMN1; SMN2ALDH1A1TP53CNR1
SCHEMBL16011202 0.80 FAAH (0.60) FAAHASAH2SMN1; SMN2SLC6A5DEGS1
SCHEMBL2058960 0.80 FAAH (0.60) FAAHASAH2SLC6A5DEGS1CETP
SCHEMBL16011422 0.80 FAAH (0.60) FAAHASAH2SMN1; SMN2SLC6A5DEGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4384508-A2 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2024-06-19 EP claimed
WO-2024031051-A1 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2024-02-08 WO claimed
US-11866723-B2 Plant virus movement proteins and methods of using same Molecular Transfer Inc. (US) 2024-01-09 US claimed
EP-4175967-A2 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation (US) 2023-05-10 EP claimed
WO-2023018990-A2 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2023-02-16 WO claimed
WO-2022006368-A2 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation (US) 2022-01-06 WO claimed
US-10968240-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2021-04-06 US claimed
US-10155780-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2018-12-18 US claimed
US-20170029448-A1 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVEDDELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2017-02-02 US claimed
EP-2912045-A2 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer, Inc. (US) 2015-09-02 EP claimed
WO-2014070687-A2 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2014-05-08 WO claimed
EP-2696678-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer, Inc. (US) 2014-02-19 EP claimed
WO-2013158127-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2013-10-24 WO claimed
EP-2015780-B1 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER INC (US) 2012-12-12 EP claimed
WO-2012142622-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2012-10-18 WO claimed
US-7915230-B2 Reagents for transfection of eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2011-03-29 US claimed
US-20090023215-A1 Novel reagents for transfection of eukaryotic cells MOLECULAR TRANSFER (US) 2009-01-22 US claimed
EP-2015780-A2 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS Molecular Transfer, Inc. (US) 2009-01-21 EP claimed
WO-2007130073-A2 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2007-11-15 WO claimed
US-12043639-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2024-07-23 US disclosed
WO-2024145435-A2 LIPID COMPOSITIONS AND METHODS FOR DELIVERY TO IMMUNE CELLS Life Technologies Corporation (US) 2024-07-04 WO disclosed
EP-4384508-A2 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2024-06-19 EP disclosed
WO-2024031051-A1 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2024-02-08 WO disclosed
US-20240000966-A1 Lipid Compositions For In Vivo Delivery Life Technologies Corporation 2024-01-04 US disclosed
WO-2024006937-A1 LIPID COMPOSITIONS FOR IN VIVO DELIVERY Life Technologies Corporation (US) 2024-01-04 WO disclosed
EP-4175967-A2 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation (US) 2023-05-10 EP disclosed
WO-2023018990-A2 LIPIDS FOR NUCLEIC ACID DELIVERY Life Technologies Corporation (US) 2023-02-16 WO disclosed
US-20220002716-A1 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation 2022-01-06 US disclosed
WO-2022006368-A2 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF Life Technologies Corporation (US) 2022-01-06 WO disclosed
US-20210323984-A1 POL YCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. 2021-10-21 US disclosed
US-11085056-B2 Transfection complexes and methods of using the same MOLECULAR TRANSFER, INC. (US) 2021-08-10 US disclosed
US-20210189433-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer Inc. 2021-06-24 US disclosed
US-10968240-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2021-04-06 US disclosed
US-10883118-B2 Agents for improved delivery of nucleic acids to eukaryotic cells Molecular Transfer Inc. (US) 2021-01-05 US disclosed
US-20190352316-A1 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2019-11-21 US disclosed
EP-2696678-B1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER INC (US) 2019-11-20 EP disclosed
US-20190264230-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer Inc. 2019-08-29 US disclosed
US-10155780-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2018-12-18 US disclosed
US-20180340188-A1 TRANSFECTION COMPLEXES AND METHODS OF USING THE SAME MOLECULAR TRANSFER, INC. (US) 2018-11-29 US disclosed
US-10138497-B2 Agents for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2018-11-27 US disclosed
US-20180237790-A1 FORMULATIONS AND COMPOSITIONS FOR DELIVERY OF NUCLEIC ACIDS TO PLANT CELLS FORREST INNOVATIONS LTD. (IL) 2018-08-23 US disclosed
EP-3334831-A1 FORMULATIONS AND COMPOSITIONS FOR DELIVERY OF NUCLEIC ACIDS TO PLANT CELLS Forrest Innovations Ltd. (IL) 2018-06-20 EP disclosed
US-20180002724-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer Inc. 2018-01-04 US disclosed
EP-2604255-B1 Novel reagents for transfection of eukaryotic cells MOLECULAR TRANSFER INC (US) 2017-10-25 EP disclosed
US-9765359-B2 Agents for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2017-09-19 US disclosed
WO-2017025967-A1 FORMULATIONS AND COMPOSITIONS FOR DELIVERY OF NUCLEIC ACIDS TO PLANT CELLS FORREST INNOVATIONS LTD. (IL) 2017-02-16 WO disclosed
US-20170029448-A1 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVEDDELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2017-02-02 US disclosed
US-20160130607-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer Inc. 2016-05-12 US disclosed
US-9259475-B2 Agents for improved delivery of nucleic acids to eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2016-02-16 US disclosed
US-20140213637-A1 Agents for Improved Delivery of Nucleic Acids to Eukaryotic Cells Molecular Transfer Inc. (US) 2014-07-31 US disclosed
US-8759499-B2 Lipids for transfection of Eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2014-06-24 US disclosed
EP-2696678-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS Molecular Transfer, Inc. (US) 2014-02-19 EP disclosed
WO-2013158127-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2013-10-24 WO disclosed
EP-2604255-A1 Novel reagents for transfection of eukaryotic cells Molecular Transfer, Inc. (US) 2013-06-19 EP disclosed
EP-2015780-B1 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER INC (US) 2012-12-12 EP disclosed
WO-2012142622-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2012-10-18 WO disclosed
US-20120052574-A1 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2012-03-01 US disclosed
US-20110200624-A1 NOVEL PEPTIDES FOR USE IN TRANSFECTION MOLECULAR TRANSFER, INC. (US) 2011-08-18 US disclosed
US-7915230-B2 Reagents for transfection of eukaryotic cells MOLECULAR TRANSFER, INC. (US) 2011-03-29 US disclosed
WO-2010014915-A2 NOVEL PEPTIDES FOR USE IN TRANSFECTION MOLECULAR TRANSFER, INC. (US) 2010-02-04 WO disclosed
US-20090023215-A1 Novel reagents for transfection of eukaryotic cells MOLECULAR TRANSFER (US) 2009-01-22 US disclosed
EP-2015780-A2 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS Molecular Transfer, Inc. (US) 2009-01-21 EP disclosed
WO-2007130073-A2 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2007-11-15 WO disclosed
WO-2007130073-A2 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS MOLECULAR TRANSFER, INC. (US) 2007-11-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (20 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180340188-A1 TRANSFECTION COMPLEXES AND METHODS OF USING THE SAME TIAL1, NPC1L1, LIPA FAAH 2128/4885ASAH2 613/4885SMN1; SMN2 4171/4885
US-12043639-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells PHOSPHO1, MBOAT7, PLTP FAAH 3332/4885ASAH2 1072/4885SMN1; SMN2 2031/4885
US-11866723-B2 Plant virus movement proteins and methods of using same HDLBP, PHAX, PLTP FAAH 3370/4885ASAH2 3573/4885SMN1; SMN2 3393/4885
US-10883118-B2 Agents for improved delivery of nucleic acids to eukaryotic cells SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-20140213637-A1 Agents for Improved Delivery of Nucleic Acids to Eukaryotic Cells SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-10968240-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells PHOSPHO1, MBOAT7, PLTP FAAH 3332/4885ASAH2 1072/4885SMN1; SMN2 2031/4885
US-10138497-B2 Agents for improved delivery of nucleic acids to eukaryotic cells SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-10155780-B2 Polycationic methyl phospholipids for improved delivery of nucleic acids to eukaryotic cells PHOSPHO1, MBOAT7, PLTP FAAH 3166/4885ASAH2 811/4885SMN1; SMN2 2830/4885
US-20240000966-A1 Lipid Compositions For In Vivo Delivery CHMP4B, LIPA, CETP FAAH 1248/4885ASAH2 72/4885SMN1; SMN2 2806/4885
US-20170029448-A1 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVEDDELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS PHOSPHO1, PLTP, MBOAT7 FAAH 3226/4885ASAH2 994/4885SMN1; SMN2 3360/4885
US-20220002716-A1 TRINUCLEOTIDE CAP ANALOGS, PREPARATION AND USES THEREOF RNGTT, RNMT, CPSF7 FAAH 4547/4885ASAH2 2798/4885SMN1; SMN2 611/4885
US-20090023215-A1 Novel reagents for transfection of eukaryotic cells FUS, PHAX, PICALM FAAH 3351/4885ASAH2 1978/4885SMN1; SMN2 2842/4885
US-11085056-B2 Transfection complexes and methods of using the same TIAL1, NPC1L1, LIPA FAAH 2128/4885ASAH2 613/4885SMN1; SMN2 4171/4885
US-20210189433-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-20190352316-A1 POLYCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS PHOSPHO1, MBOAT7, PLTP FAAH 3332/4885ASAH2 1072/4885SMN1; SMN2 2031/4885
US-20120052574-A1 NOVEL REAGENTS FOR TRANSFECTION OF EUKARYOTIC CELLS FUS, PHAX, PICALM FAAH 3351/4885ASAH2 1978/4885SMN1; SMN2 2842/4885
US-20160130607-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-20210323984-A1 POL YCATIONIC METHYL PHOSPHOLIPIDS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS POLRMT, PHOSPHO1, MBOAT7 FAAH 3358/4885ASAH2 845/4885SMN1; SMN2 2318/4885
US-20190264230-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885
US-20180002724-A1 AGENTS FOR IMPROVED DELIVERY OF NUCLEIC ACIDS TO EUKARYOTIC CELLS SNRPE, POLRMT, PHAX FAAH 3537/4885ASAH2 147/4885SMN1; SMN2 1738/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.