SCHEMBL7206793

SCHEMBL7206793

C#Cc1c[nH]c(=O)nc1NC(=O)OCC1CCCC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 8/20 0.39
MAOB P27338 5/20 0.39
MGLL Q99685 2/20 0.38
PTGIR P43119 1/20 0.36
ACHE P22303 2/20 0.34
TSHR P16473 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC3 O15379 3/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC2 Q92769 3/20 0.34
CHRM2 P08172 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
HTT P42858 1/20 0.33
NAAA Q02083 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208761 0.98 BCHE (0.39) BCHEMAOBMGLLPTGIRACHE
SCHEMBL7205752 0.95 BCHE (0.41) BCHEMAOBMGLLPTGIRACHE
SCHEMBL7206536 0.80 SMN1; SMN2 (0.39) BCHEMAOBMGLLTSHRNPC1
SCHEMBL7212661 0.78 CSNK2A2 (0.37) TSHRHTT
SCHEMBL7204740 0.76 TSHR (0.38) TSHRNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL3825844 0.76 LMNA (0.41) NPC1ALDH1A1RAB9ASMN1; SMN2NAAA
SCHEMBL7212676 0.74 RAF1 (0.33)
SCHEMBL7207482 0.73 LMNA (0.35) BCHEACHEALDH1A1RAB9ASMN1; SMN2
SCHEMBL7205833 0.73 ALDH1A1 (0.42) TSHRALDH1A1SMN1; SMN2
SCHEMBL7212657 0.72 NAAA (0.43) BCHEMGLLACHENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060183-B1 5'-DEOXYCYTIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
EP-1060183-A1 5'-DEOXYCYTIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-20 EP disclosed
WO-1999040099-A1 5'-DEOXYCYTIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-08-12 WO disclosed