SCHEMBL7363033

SCHEMBL7363033

O=C(O)CCC(c1ccccc1Cl)C1CC1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.36
OPRM1 P35372 2/20 0.35
TSHR P16473 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2D6 P10635 1/20 0.34
CPA3 P15088 1/20 0.34
NOTUM Q6P988 1/20 0.34
OPRL1 P41146 2/20 0.33
CACNA2D1 P54289 2/20 0.33
CACNA1B Q00975 2/20 0.33
CACNB1 Q02641 2/20 0.33
ACP3 P15309 1/20 0.33
FFAR1 O14842 1/20 0.33
FOLH1 Q04609 1/20 0.33
CACNA1G O43497 1/20 0.33
CACNA1C Q13936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361098 0.84 MAPK1 (0.37) CYP2C19NOTUMCACNA2D1CACNA1BCACNB1
SCHEMBL7367032 0.84 ALDH1A1 (0.36) ALDH1A1CYP1A2TSHRCYP2C19POLB
SCHEMBL7363863 0.84 CNR2 (0.36) ALDH1A1CYP1A2TSHRCYP2C19MEN1
SCHEMBL7368272 0.82 CYP2C19 (0.41) ALDH1A1CYP1A2TSHRCYP2C19CYP2D6
SCHEMBL7368286 0.82 LMNA (0.43) ALDH1A1CYP1A2TSHRPOLBCYP2D6
SCHEMBL7365442 0.80 FFAR4 (0.40) ALDH1A1CYP1A2FFAR1
SCHEMBL7399249 0.79 GABBR2 (0.39) CYP1A2TSHRCYP2C19MEN1POLB
SCHEMBL7367783 0.76 HTT (0.37) OPRM1FFAR1
SCHEMBL7369266 0.75 KDM4E (0.38) ALDH1A1MEN1POLBKMT2A
SCHEMBL7401588 0.74 NAALAD2 (0.42) ALDH1A1CYP1A2CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0771196-A4 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 1997-09-03 EP disclosed
EP-0771196-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-05-07 EP disclosed
WO-1996007405-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-03-14 WO disclosed