SCHEMBL7437102

SCHEMBL7437102

N=C(N)NC(CCCB(O)OS(=O)(=O)c1ccccc1)NC(=O)C1(C(=O)NCCc2ccc(O)cc2)CCCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.33
CA1 P00915 4/20 0.33
PLAAT3 P53816 1/20 0.32
PLAAT5 Q96KN8 1/20 0.32
PLAAT2 Q9NWW9 1/20 0.32
PLAAT4 Q9UL19 1/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
CA5A P35218 3/20 0.31
CA12 O43570 2/20 0.31
CA9 Q16790 2/20 0.31
CA4 P22748 1/20 0.31
CA7 P43166 1/20 0.31
CA14 Q9ULX7 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448384 0.92 MMP8 (0.37) MMP1MMP2MMP3SPHK1
SCHEMBL7442402 0.88 AKR1C3 (0.39) CA2CA1CA9CA7CA14
SCHEMBL7445495 0.88 USP2 (0.32) CA2CA1MMP2CA12CA9
SCHEMBL7445682 0.86 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7433244 0.84 F2 (0.34) CA2MMP1ITGB1ITGA4
SCHEMBL7433114 0.83 TBXA2R (0.30)
SCHEMBL7444716 0.83 MME (0.37) ITGB1ITGA4
SCHEMBL7429926 0.82 CA12 (0.33) CA2CA1CA12CA9ITGB1
SCHEMBL7433865 0.81 ITGB1 (0.31) ITGB1ITGA4ALDH1A1
SCHEMBL7443545 0.80 ALDH1A1 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814622-A COMPOUND USEFUL AS TRYPSIN LIKE SERINE PROTEASE AS THROMBIN INHIBITORS ADIR ET COMPAGNIE (FR) 1998-09-29 US disclosed