SCHEMBL7433244

SCHEMBL7433244

N=C(N)NC(CCCB(O)OS(=O)(=O)c1ccccc1)NC(=O)C1(C(=O)NCc2ccc3ccccc3c2)CCCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.34
F10 P00742 2/20 0.34
METAP2 P50579 1/20 0.34
METAP1 P53582 1/20 0.34
MC4R P32245 3/20 0.33
MC3R P41968 3/20 0.33
MC1R Q01726 2/20 0.33
MC5R P33032 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMB5 P28074 1/20 0.33
PSMB2 P49721 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
NPY5R Q15761 1/20 0.32
TPSAB1 Q15661 1/20 0.31
BDKRB1 P46663 2/20 0.31
BDKRB2 P30411 1/20 0.31
CA2 P00918 1/20 0.31
FAAH O00519 1/20 0.31
MMP1 P03956 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448384 0.85 MMP8 (0.37) F10MMP1
SCHEMBL7445682 0.85 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7437102 0.84 CA2 (0.33) ITGB1ITGA4CA2MMP1
SCHEMBL7445495 0.84 USP2 (0.32) F2ITGB1ITGA4TPSAB1CA2
SCHEMBL7442402 0.83 AKR1C3 (0.39) CA2
SCHEMBL7433114 0.82 TBXA2R (0.30)
SCHEMBL7444716 0.82 MME (0.37) ITGB1ITGA4
SCHEMBL7433865 0.81 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7443545 0.80 ALDH1A1 (0.42)
SCHEMBL7429926 0.79 CA12 (0.33) F2ITGB1ITGA4CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814622-A COMPOUND USEFUL AS TRYPSIN LIKE SERINE PROTEASE AS THROMBIN INHIBITORS ADIR ET COMPAGNIE (FR) 1998-09-29 US disclosed