SCHEMBL7429926

SCHEMBL7429926

CN(CCc1ccccc1)C(=O)C1(C(=O)NC(CCCB(O)OS(=O)(=O)c2ccccc2)NC(=N)N)CCCC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
F2 P00734 5/20 0.32
SPHK1 Q9NYA1 4/20 0.32
ITGB1 P05556 1/20 0.30
ITGA4 P13612 1/20 0.30
PLG P00747 2/20 0.30
PRSS1 P07477 2/20 0.30
PLAT P00750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448384 0.85 MMP8 (0.37) SPHK1PRSS1
SCHEMBL7437102 0.82 CA2 (0.33) CA12CA1CA2CA9SPHK1
SCHEMBL7433865 0.82 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7445682 0.80 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7442402 0.80 AKR1C3 (0.39) CA1CA2CA9
SCHEMBL7444716 0.79 MME (0.37) ITGB1ITGA4
SCHEMBL7445495 0.79 USP2 (0.32) CA12CA1CA2CA9F2
SCHEMBL7433244 0.79 F2 (0.34) CA2F2ITGB1ITGA4
SCHEMBL7433114 0.78 TBXA2R (0.30)
SCHEMBL7443545 0.77 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814622-A COMPOUND USEFUL AS TRYPSIN LIKE SERINE PROTEASE AS THROMBIN INHIBITORS ADIR ET COMPAGNIE (FR) 1998-09-29 US disclosed