SCHEMBL7445495

SCHEMBL7445495

N=C(N)NC(CCCB(O)OS(=O)(=O)c1ccccc1)NC(=O)C1(C(=O)NCCNS(=O)(=O)c2ccccc2)CCCC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.32
TBXA2R P21731 3/20 0.32
TBXAS1 P24557 1/20 0.32
ALDH1A1 P00352 4/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA12 O43570 1/20 0.31
MMP2 P08253 1/20 0.31
CA9 Q16790 1/20 0.31
F2 P00734 2/20 0.31
TMPRSS6 Q8IU80 2/20 0.31
PPARG P37231 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
PKM P14618 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HTT P42858 1/20 0.30
TPSAB1 Q15661 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448384 0.89 MMP8 (0.37) MMP2LMNA
SCHEMBL7437102 0.88 CA2 (0.33) ALDH1A1CA1CA2CA12MMP2
SCHEMBL7445682 0.87 ITGB1 (0.31) ITGB1ITGA4
SCHEMBL7433114 0.86 TBXA2R (0.30) TBXA2R
SCHEMBL7433244 0.84 F2 (0.34) CA2F2TPSAB1ITGB1ITGA4
SCHEMBL7442402 0.83 AKR1C3 (0.39) ALDH1A1CA1CA2CA9LMNA
SCHEMBL7444716 0.82 MME (0.37) ITGB1ITGA4
SCHEMBL7433865 0.81 ITGB1 (0.31) ALDH1A1ITGB1ITGA4
SCHEMBL7443545 0.80 ALDH1A1 (0.42) ALDH1A1HDAC3HDAC1PKM
SCHEMBL7429926 0.79 CA12 (0.33) CA1CA2CA12CA9F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814622-A COMPOUND USEFUL AS TRYPSIN LIKE SERINE PROTEASE AS THROMBIN INHIBITORS ADIR ET COMPAGNIE (FR) 1998-09-29 US disclosed