SCHEMBL75835

SCHEMBL75835

CCN1C(=O)N[C@H](CS(=O)(=O)Cl)C1=O

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
F2 P00734 1/20 0.32
ELANE P08246 1/20 0.32
CTSG P08311 1/20 0.32
CTRC Q99895 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL75836 1.00 LMNA (0.40) LMNAADORA3F2ELANECTSG
SCHEMBL22063690 0.81 LMNA (0.47) LMNAADORA3F2ELANECTSG
SCHEMBL12099135 0.81 LMNA (0.47) LMNAADORA3F2ELANECTSG
SCHEMBL74109 0.78 RIPK1 (0.38)
SCHEMBL74107 0.78 RIPK1 (0.38)
SCHEMBL1362950 0.75 LMNA (0.46) LMNAADORA3F2ELANECTSG
SCHEMBL25408450 0.73 LMNA (0.49) LMNAADORA3F2ELANECTSG
SCHEMBL7751272 0.73 LMNA (0.44) LMNAADORA3F2ELANECTSG
SCHEMBL8716129 0.68 ALDH1A1 (0.40) LMNAADORA3
SCHEMBL4748698 0.66 LMNA (0.48) LMNAADORA3F2ELANECTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129412-B2 Hydantoin derivatives useful as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2012-03-06 US disclosed
EP-1828166-B1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2009-07-22 EP disclosed
US-20080280950-A1 Hydantoin Derivatives Useful as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-11-13 US disclosed
EP-1828166-A1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS AstraZeneca AB (SE) 2007-09-05 EP disclosed
WO-2006064218-A1 HYDANTOIN DERIVATIVES USEFUL AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2006-06-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280950-A1 Hydantoin Derivatives Useful as Metalloproteinase Inhibitors MMP3, MMP9, MMP2 LMNA 1052/4885ADORA3 2071/4885F2 330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.