SCHEMBL7696757

SCHEMBL7696757

COc1ccc2c(c1)c(CC(=O)O)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 2/20 0.69
AKR1C3 P42330 4/20 0.67
AKR1C4 P17516 2/20 0.67
PTGS1 P23219 2/20 0.67
AKR1C2 P52895 2/20 0.67
PPARD Q03181 3/20 0.64
PPARG P37231 3/20 0.64
PPARA Q07869 2/20 0.64
LMNA P02545 5/20 0.61
ALDH1A1 P00352 3/20 0.61
MEN1 O00255 2/20 0.61
CYP1A2 P05177 2/20 0.61
MAPT P10636 2/20 0.61
CYP2C9 P11712 2/20 0.61
PMP22 Q01453 2/20 0.61
KMT2A Q03164 2/20 0.61
HIF1A Q16665 2/20 0.61
RGS12 O14924 1/20 0.61
CYP3A4 P08684 1/20 0.61
PKM P14618 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20769739 0.91 PLA2G2A (0.83) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL3030239 0.89 MTNR1A (0.61) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL11332785 0.87 MTNR1A (0.59) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL20769719 0.86 ALDH1A1 (0.65) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL7053553 0.84 CACNB4 (0.62) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL8171657 0.82 KEAP1 (0.57) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL10946754 0.82 AKR1C3 (0.69) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2
SCHEMBL7692305 0.82 CHRM1 (0.65) PLA2G2APPARDPPARGPPARALMNA
SCHEMBL7963252 0.81 PLA2G2A (1.00) PLA2G2APPARDPPARGPPARALMNA
Methoxyacetic Acid SCHEMBL9738426 0.81 LMNA (0.55) PLA2G2AAKR1C3AKR1C4PTGS1AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002020478-A1 N-BENZYLINDOLE-3-ACETIC ACID DERIVATIVES FOR USE IN THE TREATMENT OF DRUG RESISTAN CANCER DUBLIN CITY UNIVERSITY (IE) 2002-03-14 WO claimed
WO-2002020478-A1 N-BENZYLINDOLE-3-ACETIC ACID DERIVATIVES FOR USE IN THE TREATMENT OF DRUG RESISTAN CANCER DUBLIN CITY UNIVERSITY (IE) 2002-03-14 WO disclosed