SCHEMBL7698169

SCHEMBL7698169

N#Cc1cc(F)c(-n2ccc(C(F)(F)F)cc2=O)cc1F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 6/20 0.38
BCAT2 O15382 7/20 0.36
BCAT1 P54687 7/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
CTSK P43235 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984454 0.85 BCAT1 (0.42) BCAT2BCAT1
SCHEMBL7695435 0.80 PGR (0.40) BCAT2BCAT1ALDH1A1
SCHEMBL7085889 0.75 TRPV4 (0.37) TRPV4BCAT2BCAT1CYP11B1CYP11B2
SCHEMBL7753821 0.75 CYP11B1 (0.41) TRPV4BCAT2BCAT1CYP11B1CYP11B2
SCHEMBL9599435 0.73 ESR1 (0.43) KDM4EALDH1A1GAA
SCHEMBL9598055 0.73 SMN1; SMN2 (0.41) KDM4EALDH1A1GAA
SCHEMBL9730810 0.72 GABRB3 (0.37) TRPV4KDM4EALDH1A1GAA
SCHEMBL10679727 0.70 CA2 (0.36) GAA
SCHEMBL11954634 0.69 ALK (0.47) TRPV4ALDH1A1
SCHEMBL9598871 0.69 ALDH1A1 (0.48) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002020487-A1 SUBSTITUTED 1-ARYL-PYRIDIN-2-(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 2002-03-14 WO disclosed