Brl-15,572

Brl-15,572

SCHEMBL7741355

OC(CN1CCN(c2cccc(Cl)c2)CC1)C(c1ccccc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 1.00
KMT2A Q03164 4/20 1.00
TSHR P16473 2/20 1.00
MAPT P10636 2/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2D6 P10635 1/20 1.00
ALOX15 P16050 1/20 1.00
CYP2C19 P33261 1/20 1.00
HIF1A Q16665 1/20 1.00
LMNA P02545 2/20 0.97
NPSR1 Q6W5P4 2/20 0.97
GMNN O75496 1/20 0.97
BLM P54132 1/20 0.97
PMP22 Q01453 1/20 0.97
IGF1R P08069 1/20 0.61
RECQL P46063 2/20 0.59
SIGMAR1 Q99720 2/20 0.55
MAPK1 P28482 1/20 0.55
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brl-15,572 SCHEMBL17978413 0.99 MEN1 (1.00) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL8944148 0.87 IGF1R (0.79) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL6017439 0.87 KMT2A (0.76) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL19852034 0.77 RECQL (0.87) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL30001848 0.77 RECQL (0.87) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL17207530 0.76 POLB (0.65) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL4355715 0.76 MEN1 (0.62) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL27959848 0.76 IGF1R (1.00) MEN1KMT2ATSHRMAPTCYP1A2
SCHEMBL9646111 0.75 ALDH1A1 (0.73) MEN1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL9374413 0.75 SIGMAR1 (0.76) TSHRMAPTLMNASIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
CN-117899219-A Application of HTR1D as target spot in medicine for treating pain-depression co-diseases 徐州医科大学 2024-04-19 CN claimed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO claimed
US-20220146492-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY SHINE IAN BASIL (US) 2022-05-12 US claimed
EP-3953000-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY Shine, Ian Basil (US) 2022-02-16 EP claimed
EP-3160464-A1 USE OF BUSPIRONE METABOLITES Contera Pharma APS (DK) 2017-05-03 EP claimed
WO-2015197079-A1 USE OF BUSPIRONE METABOLITES CONTERA PHARMA APS (DK) 2015-12-30 WO claimed
US-20260083706-A1 5HT AGONISTS FOR TREATING DISORDERS UNIV CALIFORNIA (US) 2026-03-26 US disclosed
EP-4696377-A2 5HT AGONISTS FOR TREATING DISORDERS The Regents of the University of California (US) 2026-02-18 EP disclosed
US-12551481-B2 Molecular targets for addiction THE JACKSON LABORATORY (US) 2026-02-17 US disclosed
CN-116891405-B Chiral alpha, alpha-diaryl ketone compound and preparation method and application thereof 五邑大学 2025-12-05 CN disclosed
EP-4043016-B1 THE 5HT AGONIST CLEMIZOLE FOR USE IN TREATING EPILEPSY DISORDERS UNIV CALIFORNIA (US) 2025-10-29 EP disclosed
US-12447144-B2 5HT agonists for treating disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-10-21 US disclosed
US-20140221385-A1 COMBINATIONS OF SEROTONIN RECEPTOR AGONISTS FOR TREATMENT OF MOVEMENT DISORDERS CONCIT PHARMA APS (DK) 2014-08-07 US disclosed
US-8569481-B2 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions PHARMACEUTICALS, INC. (US) 2013-10-29 US disclosed
WO-2012163365-A1 COMBINATIONS OF SEROTONIN RECEPTOR AGONISTS FOR TREATMENT OF MOVEMENT DISORDERS CONCIT PHARMA APS (DK) 2012-12-06 WO disclosed
US-20110118136-A1 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions KOESTER HUBERT 2011-05-19 US disclosed
US-20100298168-A1 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions HK PHARMACEUTICALS, INC. 2010-11-25 US disclosed
US-20100248264-A1 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions HK PHARMACEUTICALS, INC. 2010-09-30 US disclosed
WO-2001015677-A2 USE OF 5-HT1B/1D AGONISTS TO TREAT OTIC PAIN ALCON LABORATORIES, INC. (US) 2001-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118136-A1 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions PTMS, QPCTL, SRMS MEN1 3426/4885KMT2A 2736/4885TSHR 3135/4885
US-20260083706-A1 5HT AGONISTS FOR TREATING DISORDERS SLC6A4, SLC6A2, TPH2 MEN1 951/4885KMT2A 1017/4885TSHR 419/4885
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS HTR2A, HTR5A, HTR6 MEN1 2593/4885KMT2A 1760/4885TSHR 417/4885
US-12447144-B2 5HT agonists for treating disorders HTR1A, HTR5A, HTR2A MEN1 901/4885KMT2A 1091/4885TSHR 384/4885
US-20100298168-A1 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions CHLSN, PTMS, SRMS MEN1 2224/4885KMT2A 4241/4885TSHR 4673/4885
US-12551481-B2 Molecular targets for addiction HTR1D, HTR2A, HTR1A MEN1 3653/4885KMT2A 667/4885TSHR 503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.