SCHEMBL7743750

SCHEMBL7743750

CC(C)(C)c1ccc([O-])c(C(C)(C)C)c1.[Na+]

nearest known ligand 0.41

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 2/20 0.32
CA2 known ✓ P00918 2/20 0.32
CA12 known ✓ O43570 1/20 0.32
ALDH1A1 P00352 6/20 0.41
ALOX15 P16050 2/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NR1I2 O75469 1/20 0.41
MAPT P10636 3/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
RECQL P46063 1/20 0.38
KMT2A Q03164 1/20 0.38
TSHR P16473 1/20 0.37
LMNA P02545 1/20 0.36
TYR P14679 1/20 0.36
NPC1 O15118 1/20 0.35
PLA2G1B P04054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL7746261 0.95 ALDH1A1 (0.41) ALDH1A1ALOX15HPGDHSD17B10TDP1
Lithium Ion SCHEMBL7743747 0.95 ALDH1A1 (0.41) ALDH1A1ALOX15HPGDHSD17B10TDP1
SCHEMBL10874622 0.95 ALDH1A1 (0.41) ALDH1A1ALOX15HPGDHSD17B10TDP1
SCHEMBL5396186 0.95 ALDH1A1 (0.41) ALDH1A1ALOX15HPGDHSD17B10TDP1
Hydrochloric Acid SCHEMBL6039934 0.93 ALDH1A1 (0.40) ALDH1A1ALOX15HPGDHSD17B10TDP1
SCHEMBL5679072 0.93 ALDH1A1 (0.40) ALDH1A1ALOX15HPGDHSD17B10TDP1
SCHEMBL4363292 0.90 ALDH1A1 (0.38) ALDH1A1ALOX15HPGDHSD17B10TDP1
Phosphoric Acid SCHEMBL29534935 0.89 NR1I2 (0.39) ALDH1A1ALOX15HPGDHSD17B10TDP1
Phosphoric Acid SCHEMBL27702683 0.89 NR1I2 (0.39) ALDH1A1ALOX15HPGDHSD17B10TDP1
SCHEMBL1451091 0.85 ALDH1A1 (0.34) ALDH1A1ALOX15HPGDHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102827205-A Preparation method of nucleating agent CHINA PETROLEUM & CHEMICAL 2012-12-19 CN disclosed
CN-102807474-A Preparation methods of substituted diaryl phenol, organophosphorus ester and organic phosphate CHINA PETROLEUM & CHEMICAL 2012-12-05 CN disclosed
CN-101942126-B Transparent antistatic polyethylene film master batch PETROCHINA CO LTD 2012-08-08 CN disclosed
CN-102408444-A Ultrasonic preparation method of fine transparent nucleating agent CHINA PETROLEUM & CHEMICAL 2012-04-11 CN disclosed
CN-102382359-A Preparation method of ultrafine organic phosphate nucleating agent CHINA PETROLEUM & CHEMICAL 2012-03-21 CN disclosed
CN-102382135-A Preparation method of organic phosphate polypropylene nucleating agent CHINA PETROLEUM & CHEMICAL 2012-03-21 CN disclosed
US-6429273-B1 ANIONIC POLYMERIZATION OF STYRENE USING MAGNESIUM AND ALKALI METAL-BASED INITIATORS; CONTROLLED MOLECULAR WEIGHT DISTRIBUTION; CONTROLLABLE RATE PREVENTS RUNAWAY REACTION; EXCELLENT MOLDING CHARACTERISTICS ASAHI KASEI KABUSHIKI KAISHA (JP) 2002-08-06 US disclosed
CN-1319584-A Process for preparing 3,5-di-tert-butyl salicylic acid HUBEI INST OF CHEMISTRY (CN) 2001-10-31 CN disclosed