SCHEMBL7765362

SCHEMBL7765362

O=C1N=C(c2ccccc2)CO1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.56
ALDH1A1 P00352 4/20 0.56
KDM4E B2RXH2 4/20 0.56
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
LMNA P02545 3/20 0.56
GAA P10253 2/20 0.56
DHFR P00374 1/20 0.49
KMT2A Q03164 3/20 0.44
AXL P30530 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
ALOX12 P18054 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
PDE3B Q13370 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31541474 0.80 ALDH1A1 (0.41) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL1570052 0.80 MAPT (0.37) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL28684618 0.80 NPC1 (0.46) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL28932271 0.80 NPC1 (0.50) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL31541475 0.80 ALDH1A1 (0.41) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL11719543 0.78 PDE3B (0.49) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL28703819 0.78 CHRNB4 (0.45) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL28677904 0.78 PDE3B (0.51) PDE3BPDE3APTGS1CHRNB4CHRNA3
SCHEMBL28687865 0.78 CHRNB4 (0.45) MAPTKDM4ENPC1RAB9AKMT2A
SCHEMBL28677905 0.78 PDE3B (0.49) MAPTALDH1A1KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119404851-A Antibacterial application of indolizine-spiro-oxazolinone compound 青岛农业大学 2025-02-11 CN claimed
CN-118393827-A High-temperature-resistant low-corrosion photoresist stripping liquid and preparation method and application thereof 浙江奥首材料科技有限公司 2024-07-26 CN claimed
CN-119404851-A Antibacterial application of indolizine-spiro-oxazolinone compound 青岛农业大学 2025-02-11 CN disclosed
CN-118393827-A High-temperature-resistant low-corrosion photoresist stripping liquid and preparation method and application thereof 浙江奥首材料科技有限公司 2024-07-26 CN disclosed
CN-113999131-B Method for preparing amide derivative by amination of alkyl C-H bond under catalysis of nickel promoted by visible light 苏州大学 2022-06-28 CN disclosed
CN-113999131-A Method for preparing amide derivative by amination of alkyl C-H bond under catalysis of nickel promoted by visible light 苏州大学 2022-02-01 CN disclosed
US-10100053-B2 Process for the preparation of 8-(4-aminophenoxy)-4H-pyrido[2,3-b]pyrazin-3-one derivatives CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-10-16 US disclosed
US-9796675-B1 Intermediate for synthesizing paroxetine, method for preparing the same, and uses thereof ZHEJIANG JIUZHOU PHARMACEUTICAL CO., LTD (CN) 2017-10-24 US disclosed
US-20170298065-A1 PROCESS FOR THE PREPARATION OF 8-(4-AMINOPHENOXY)-4H-PYRIDO[2,3-B]PYRAZIN-3-ONE DERIVATIVES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2017-10-19 US disclosed
US-20170283380-A1 Intermediate for Synthesizing Paroxetine, Method for Preparing the same, and Uses Thereof ZHEJIANG JIUZHOU PHARM CO LTD (CN) 2017-10-05 US disclosed
EP-3199526-A1 INTERMEDIATE FOR USE IN SYNTHESIZING PAROXETINE, PREPARATION METHOD FOR THE INTERMEDIATE, AND USES THEREOF Zhejiang Jiuzhou Pharmaceutical Co., Ltd (CN) 2017-08-02 EP disclosed
WO-2016016865-A1 A PROCESS FOR THE PREPARATION OF NUCLEOSIDE PHOSPHORAMIDATE LUPIN LIMITED (IN) 2016-02-04 WO disclosed
EP-0859766-B1 CHIRAL METHYL PHENYL OXAZOLIDINONES SCHERING AG (DE) 2001-05-16 EP disclosed
EP-0859766-A1 CHIRAL METHYL PHENYL OXAZOLIDINONES SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-26 EP disclosed
WO-1997015561-A1 CHIRAL METHYL PHENYL OXAZOLIDINONES SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10100053-B2 Process for the preparation of 8-(4-aminophenoxy)-4H-pyrido[2,3-b]pyrazin-3-one derivatives PAM, PDXK, GRHPR MAPT 2753/4885ALDH1A1 1647/4885KDM4E 377/4885
US-20170283380-A1 Intermediate for Synthesizing Paroxetine, Method for Preparing the same, and Uses Thereof TPH2, TPH1, HTR1F MAPT 3006/4885ALDH1A1 1943/4885KDM4E 1638/4885
US-20170298065-A1 PROCESS FOR THE PREPARATION OF 8-(4-AMINOPHENOXY)-4H-PYRIDO[2,3-B]PYRAZIN-3-ONE DERIVATIVES TDO2, HPD, PDXK MAPT 3185/4885ALDH1A1 879/4885KDM4E 58/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.