SCHEMBL7790448

SCHEMBL7790448

OCC[N]c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.43
HTR3E A5X5Y0 3/20 0.43
HTR3B O95264 3/20 0.43
HTR3D Q70Z44 3/20 0.43
HTR3C Q8WXA8 3/20 0.43
SLC22A2 O15244 2/20 0.43
SLC22A1 O15245 2/20 0.43
SLC22A3 O75751 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
PLAU P00749 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 2/20 0.38
CYP2A6 P11509 1/20 0.38
NOS3 P29474 4/20 0.37
NOS1 P29475 4/20 0.37
NOS2 P35228 4/20 0.37
ALDH1A1 P00352 3/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5490413 0.87 ADRA2A (0.32) NOS3NOS1ADRA2AADRA2BADRA2C
SCHEMBL7794049 0.85 HTR3A (0.39) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL10990336 0.78 LMNA (0.40) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7789999 0.76 HTR3E (0.43) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL1720891 0.75 ALDH1A1 (0.41) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8696375 0.74 HTR3E (0.50) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL1735291 0.70 NOS3 (0.44) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7840304 0.66 ALDH1A1 (0.33) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL3282366 0.64 LMNA (0.57) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL3282369 0.64 LMNA (0.57) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed
US-H533-H 1H-PYRAZOLO(1,5-B)OR(5,1-C)-1,2,4-TRIAZOLE MAGENTA COUPLER FUJI PHOTO FILM CO., LTD. (JP) 1988-10-04 US disclosed
US-4256896-A THIAZOLE, IMIDAZOLINE, AND OXAZOLINE DYES; DISPERSE DYES; ANIONIC DYES; TEXTILES CIBA-GEIGY AKTIENGESELLSCHAFT (DE) 1981-03-17 US disclosed
US-4246422-A Naphtholactam dyestuffs CIBA-GEIGY AG (CH) 1981-01-20 US disclosed
US-4246410-A BENZINDOLE DYES OF YELLOW AND RED CIBA -GEIGY AKTIENGESELLSCHAFT (CH) 1981-01-20 US disclosed
US-4236007-A YELLOW SHADES ON POLYESTERS CIBA-GEIGY AKTIENGESELLSCHAFT (CH) 1980-11-25 US disclosed
US-4180665-A Substituted 3-benz(cd)indol-2-(1H)-ylidene-furo[2,3-b]quinoxalin-2(3H)one dyestuffs CIBA-GEIGY AKTIENGESELLSCHAFT (CH) 1979-12-25 US disclosed
US-4148805-A POLYESTERS, RED, YELLLOW CIBA-GEIGY AG (CH) 1979-04-10 US disclosed
US-4146541-A YELLOW SHADE ON POLYESTERS CIBA-GEIGY AG (CH) 1979-03-27 US disclosed