SCHEMBL7794049

SCHEMBL7794049

OCCCC[N]c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.39
HTR3E A5X5Y0 3/20 0.39
HTR3B O95264 3/20 0.39
HTR3D Q70Z44 3/20 0.39
HTR3C Q8WXA8 3/20 0.39
SLC22A2 O15244 2/20 0.39
SLC22A1 O15245 2/20 0.39
SLC22A3 O75751 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
PLAU P00749 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
LMNA P02545 3/20 0.37
GBA1 P04062 2/20 0.37
TP53 P04637 2/20 0.37
CYP3A4 P08684 2/20 0.37
ALOX15 P16050 2/20 0.37
MAPK1 P28482 2/20 0.37
MC4R P32245 2/20 0.37
RAD52 P43351 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790448 0.85 HTR3A (0.43) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7790019 0.79 HTR3E (0.39) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7793217 0.79 HTR3E (0.44) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL10990336 0.78 LMNA (0.40) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL10503151 0.77 MIF (0.35) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7790485 0.73 ITGB3 (0.41) LMNATP53ALOX15MAPK1CYP1A2
SCHEMBL5490413 0.71 ADRA2A (0.32) ADRA2AADRA2BADRA2CNOS3NOS1
SCHEMBL10502034 0.71 ALDH1A1 (0.38) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL6651377 0.68 PLG (0.40) LMNAMAPTNOS3NOS1NOS2
SCHEMBL1803684 0.67 IGF1R (0.59) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed