Piperidine

Piperidine

SCHEMBL781392

C1CCNCC1.C1CCNCC1.O

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Piperidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4A known ✓ P27815 1/20 0.46
KDR known ✓ P35968 1/20 0.46
ALDH1A1 P00352 1/20 0.90
CXCR4 P61073 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HIF1A Q16665 1/20 0.46
MAPT P10636 1/20 0.46
CA2 P00918 1/20 0.30
CHKA P35790 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL27684596 1.00 ALDH1A1 (0.90) ALDH1A1CXCR4SMN1; SMN2HIF1AMAPT
Piperidine SCHEMBL7575332 1.00
Azepane SCHEMBL20563677 1.00
Water SCHEMBL27684593 1.00 ALDH1A1 (0.90) ALDH1A1CXCR4SMN1; SMN2HIF1AMAPT
Piperidine SCHEMBL4616564 1.00
Piperidine SCHEMBL7575329 1.00 ALDH1A1 (0.90) ALDH1A1CXCR4SMN1; SMN2HIF1AMAPT
Piperidine SCHEMBL28700802 1.00 ALDH1A1 (0.90) ALDH1A1CXCR4SMN1; SMN2HIF1AMAPT
Azepane SCHEMBL29258022 0.95
Piperidine SCHEMBL9028300 0.95
Piperidine SCHEMBL30996101 0.95 ALDH1A1 (0.82) ALDH1A1CXCR4SMN1; SMN2HIF1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 89 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023139322-A1 HYDROSILYLATION PROCESS PHOTOCATALYSED BY A MANGANESE COMPLEX ELKEM SILICONES FRANCE SAS (FR) 2023-07-27 WO claimed
EP-2935286-B1 HYDROSILYLATION METHOD ELKEM SILICONES FRANCE SAS (FR) 2018-08-01 EP claimed
EP-0886520-A1 CAFFEINE AND CLEMASTINE FOR TREATING RESPIRATORY DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1998-12-30 EP claimed
EP-0841947-A1 COMPOSITIONS CONTAINING ANALGESICS AND ANTIHISTAMINES AND METHODS FOR TREATING RESPIRATORY DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1998-05-20 EP claimed
WO-1997032586-A1 CAFFEINE AND CLEMASTINE FOR TREATING RESPIRATORY DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1997-09-12 WO claimed
US-5648358-A CAFFEINE AND PYRROLIDINE OR PIPERIDINE ETHER ANTIHISTAMINE PROCTER & GAMBLE COMPANY, THE 1997-07-15 US claimed
WO-1997004808-A1 COMPOSITIONS CONTAINING ANALGESICS AND ANTIHISTAMINES AND METHODS FOR TREATING RESPIRATORY DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1997-02-13 WO claimed
JP-4356462-A None JP disclosed
WO-2024146993-A1 HYDROSILYLATION PROCESS CATALYSED BY A MANGANESE COMPLEX ELKEM SILICONES FRANCE SAS (FR) 2024-07-11 WO disclosed
US-11964973-B2 Substituted bicyclic compounds useful as T cell activators BRISTOL-MYERS SQUIBB COMPANY (US) 2024-04-23 US disclosed
CN-111936231-B Nanoparticles of zero-valent metal CO complexes useful as hydrosilylation and dehydrogenative silylation catalysts 埃肯有机硅法国有限公司 2023-10-27 CN disclosed
US-20230264183-A1 NANOPARTICLES OF CO COMPLEXES OF ZERO-VALENT METALS THAT CAN BE USED AS HYDROSILYLATION AND DEHYDROGENATIVE SILYLATION CATALYSTS ELKEM SILICONES FRANCE SAS (FR) 2023-08-24 US disclosed
WO-2023139322-A1 HYDROSILYLATION PROCESS PHOTOCATALYSED BY A MANGANESE COMPLEX ELKEM SILICONES FRANCE SAS (FR) 2023-07-27 WO disclosed
US-5169855-A PIPERIDINE ETHER DERIVATIVES AS PSYCHOTROPIC DRUGS OR PLANT FUNGICIDES DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-12-08 US disclosed
US-5169855-A PIPERIDINE ETHER DERIVATIVES AS PSYCHOTROPIC DRUGS OR PLANT FUNGICIDES DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-12-08 US disclosed
CN-1058399-A New piperidine ether and thioether as cholesteral biosynthesis inhibitor MERRELL DOW PHARMA (US) 1992-02-05 CN disclosed
CN-1058399-A New piperidine ether and thioether as cholesteral biosynthesis inhibitor MERRELL DOW PHARMA (US) 1992-02-05 CN disclosed
EP-0449187-A2 Piperidin ether derivatives as psychotropic drugs or plant fungicides THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-10-02 EP disclosed
EP-0449187-A2 Piperidin ether derivatives as psychotropic drugs or plant fungicides THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-10-02 EP disclosed
US-3862158-A PIPERIDINE ETHERS HOFFMANN LA ROCHE 1975-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11964973-B2 Substituted bicyclic compounds useful as T cell activators DGKA, DGKZ, DGKK PDE4A 1415/4885KDR 2426/4885ALDH1A1 4765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.