SCHEMBL7962741

SCHEMBL7962741

OC(CCOc1ccc2cccnc2c1)N1CCC(O)(c2cnc3ccccc3n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.42
CYP3A4 P08684 1/20 0.39
DRD3 P35462 1/20 0.36
DRD2 P14416 2/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
PDE2A O00408 1/20 0.35
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALOX5AP P20292 2/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7953284 0.87 PDE10A (0.40) PDE10ACYP3A4DRD3DRD2OPRM1
SCHEMBL7962207 0.84 ALDH1A1 (0.43) DRD3DRD2OPRM1OPRD1OPRK1
SCHEMBL7962696 0.84 LTA4H (0.35) OPRM1OPRD1OPRK1OPRL1NPC1
SCHEMBL7962746 0.82 SMN1; SMN2 (0.47) PDE10AMAPTHTT
SCHEMBL7962978 0.81 PPARG (0.39) PDE10AOPRM1OPRD1OPRK1OPRL1
SCHEMBL7962748 0.81 PDE10A (0.39) PDE10ACYP3A4DRD3DRD2OPRL1
SCHEMBL7200716 0.78 KDM4E (0.38) DRD3OPRM1OPRD1OPRK1OPRL1
Sulfuric Acid SCHEMBL7968955 0.78 THRB (0.36) DRD3DRD2OPRM1HTT
SCHEMBL7965112 0.77 LMNA (0.39) OPRM1OPRD1NPC1MAPTRAB9A
Heptanoate SCHEMBL7966354 0.74 LTA4H (0.38) DRD3DRD2OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed