SCHEMBL7962207

SCHEMBL7962207

COc1cccc(OCCC(O)N2CCC(O)(c3cnc4ccccc4n3)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
MAPT P10636 5/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
TP53 P04637 6/20 0.39
THRB P10828 1/20 0.38
TSHR P16473 2/20 0.37
MAPK1 P28482 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
KDM4E B2RXH2 2/20 0.37
FGFR2 P21802 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963015 0.86 OPRM1 (0.44) ALDH1A1MAPTNPC1RAB9AOPRM1
SCHEMBL7962696 0.84 LTA4H (0.35) ALDH1A1MAPTNPC1RAB9AOPRM1
SCHEMBL7962741 0.84 PDE10A (0.42) MAPTNPC1RAB9AOPRM1OPRD1
SCHEMBL7962212 0.81 ALDH1A1 (0.41) ALDH1A1MAPTNPC1RAB9AOPRM1
SCHEMBL7965112 0.79 LMNA (0.39) ALDH1A1MAPTNPC1RAB9AOPRM1
Sulfuric Acid SCHEMBL7968955 0.79 THRB (0.36) OPRM1DRD2DRD3THRB
Heptanoate SCHEMBL7966354 0.78 LTA4H (0.38) ALDH1A1MAPTNPC1RAB9AOPRM1
SCHEMBL7963392 0.78 ADRB2 (0.35) OPRM1OPRD1OPRK1OPRL1TP53
SCHEMBL7953343 0.78 ALDH1A1 (0.46) ALDH1A1MAPTNPC1RAB9AOPRM1
Fumaric Acid SCHEMBL7966209 0.76 MAPT (0.38) ALDH1A1MAPTNPC1DRD2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
WO-2000006166-A1 5-HT1F ANTAGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed