SCHEMBL7986731

SCHEMBL7986731

COC(=O)c1cccc2c1c(-c1cncc(-c3cccc(OC)c3)c1)cn2C(C)C1CCCNC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.41
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38
TYRO3 Q06418 2/20 0.38
ABL1 P00519 1/20 0.37
EGFR P00533 1/20 0.37
SRC P12931 1/20 0.37
ABL2 P42684 1/20 0.37
CYP2C19 P33261 1/20 0.37
NEK1 Q96PY6 1/20 0.37
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
JAK2 O60674 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
AXL P30530 1/20 0.35
FLT3 P36888 1/20 0.35
MERTK Q12866 1/20 0.35
F10 P00742 1/20 0.34
DGAT2 Q96PD7 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7511168 0.93 CHEK1 (0.40) CHEK1GRIN1GRIN2BTYRO3CCNC
SCHEMBL7506739 0.92 CDK7 (0.39) CHEK1AXLF10
SCHEMBL7994754 0.91 CHEK1 (0.38) CHEK1
SCHEMBL7994227 0.89 CDK9 (0.39) CHEK1CCNCCDK8
SCHEMBL7508016 0.87 OPRK1 (0.42) CHEK1ITGB3ITGA2BAXL
SCHEMBL7990422 0.87 ABL1 (0.38) CHEK1ABL1EGFRSRCABL2
SCHEMBL7976272 0.84 CCNT1 (0.41) CHEK1ABL1EGFRSRCABL2
SCHEMBL7975970 0.82 HTR6 (0.39) CHEK1TYRO3ABL1EGFRSRC
SCHEMBL7994923 0.80 PRKCA (0.40) CHEK1TYRO3ABL1EGFRSRC
SCHEMBL7990984 0.80 CCNT1 (0.36) CHEK1TYRO3ABL1EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed