SCHEMBL7994940

SCHEMBL7994940

O=C1c2nc3nonc3nc2-c2cccc(OCc3cccnc3)c21

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.52
PRKDC P78527 5/20 0.41
HTR1A P08908 2/20 0.41
DRD2 P14416 2/20 0.41
BRD4 O60885 1/20 0.41
IKBKB O14920 1/20 0.39
SGMS2 Q8NHU3 1/20 0.38
PIK3CD O00329 1/20 0.37
PIM1 P11309 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR6 P50406 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
CGAS Q8N884 1/20 0.36
GCK P35557 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7996801 0.92 PTGES (0.52) PTGESPRKDCHTR1ADRD2BRD4
SCHEMBL7996575 0.88 PTGES (0.55) PTGESPRKDCBRD4IKBKBSGMS2
SCHEMBL7984832 0.88 PTGES (0.63) PTGESBRD4SGMS2
SCHEMBL7994971 0.80 PTGES (0.59) PTGESPRKDCHTR1ADRD2BRD4
SCHEMBL7996440 0.78 PTGES (0.54) PTGESPIK3CDCYP1A2CYP3A4ALDH1A1
SCHEMBL7984763 0.78 PTGES (0.54) PTGESALDH1A1POLB
SCHEMBL7984591 0.75 PTGES (0.61) PTGESALDH1A1POLB
SCHEMBL7996719 0.75 PTGES (0.64) PTGESPIM1ALDH1A1
SCHEMBL8339083 0.73 SGMS2 (0.48) PRKDCHTR1ADRD2BRD4IKBKB
SCHEMBL7994951 0.71 PTGES (0.56) PTGESALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO claimed
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO disclosed