SCHEMBL8002272

SCHEMBL8002272

Fc1c(F)c(F)c([B-](Cc2ccccc2)(c2c(F)c(F)c(F)c(F)c2F)c2c(F)c(F)c(F)c(F)c2F)c(F)c1F.[Na+]

nearest known ligand 0.37

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.37
TSHR P16473 5/20 0.35
CALM1 P0DP23 1/20 0.35
ALDH1A1 P00352 2/20 0.32
LOXL2 Q9Y4K0 2/20 0.32
IDO1 P14902 1/20 0.32
TRPA1 O75762 1/20 0.32
FAAH O00519 1/20 0.31
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
ELANE P08246 1/20 0.31
PRTN3 P24158 1/20 0.31
PRSS3 P35030 1/20 0.31
MAOB P27338 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929654 0.98 TP53 (0.39) TP53TSHRCALM1ALDH1A1LOXL2
Tetraphenylphosphonium SCHEMBL21750877 0.87 TP53 (0.31) TP53TSHR
SCHEMBL7980580 0.87 TP53 (0.31) TP53TSHR
SCHEMBL21750947 0.85 TP53 (0.31) TP53CYP2A6TAAR1
Tetrabuthylammonium SCHEMBL21750880 0.80 DNM1 (0.41) TP53KMT2ASMN1; SMN2
Quinoline SCHEMBL21751032 0.79
SCHEMBL21750989 0.78 KDM4E (0.38) TP53ALDH1A1KMT2ASMN1; SMN2
SCHEMBL21750875 0.77 CHRM2 (0.44) TP53TSHRALOX12KMT2AHTR2A
SCHEMBL21750997 0.75 ACHE (0.52) ALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL21750879 0.75 ACHE (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200062783-A1 PHOTO LEWIS ACID GENERATOR NIPPON SHOKUBAI CO., LTD. (JP) 2020-02-27 US disclosed
US-6100414-A Cyclopentadienyl transition metal compounds useful as polymerization catalysts EASTMAN CHEMICAL COMPANY (US) 2000-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200062783-A1 PHOTO LEWIS ACID GENERATOR LEO1, LRRK2, LSG1 TP53 2208/4885TSHR 2934/4885CALM1 3859/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.