SCHEMBL8043693

SCHEMBL8043693

Cn1cnnc1Sc1ncc(S(C)(=O)=O)s1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIP4K2C Q8TBX8 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 3/20 0.36
KDM4E B2RXH2 3/20 0.36
GCK P35557 5/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
CASP6 P55212 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LMNA P02545 1/20 0.32
USP2 O75604 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
HBB P68871 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050654 0.79 NPC1 (0.36) SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL8046664 0.79 CA12 (0.42) PIP4K2CALDH1A1HTTSMN1; SMN2HSD17B10
SCHEMBL8047637 0.78 LMNA (0.39) PIP4K2CALDH1A1HTTSMN1; SMN2HSD17B10
SCHEMBL8033687 0.76 RXRA (0.43) ALDH1A1SMN1; SMN2HSD17B10KDM4EGCK
SCHEMBL8048372 0.76 MEN1 (0.33) MEN1KMT2A
SCHEMBL7823341 0.75 TDP1 (0.56) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL8045938 0.75 HSD17B10 (0.40) ALDH1A1HTTSMN1; SMN2HSD17B10MEN1
SCHEMBL8041836 0.74 ALDH1A1 (0.42) ALDH1A1HTTSMN1; SMN2HSD17B10MEN1
SCHEMBL8045587 0.73
SCHEMBL8048331 0.73 ALDH1A1 (0.33) ALDH1A1SMN1; SMN2MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed