SCHEMBL8086489

SCHEMBL8086489

CCCN(CCC)S(=O)(=O)N(CCc1ccc([N+](=O)[O-])cc1)C(=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
CA12 O43570 3/20 0.45
CA9 Q16790 2/20 0.45
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
KCNH2 Q12809 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CA1 P00915 2/20 0.40
BMP1 P13497 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092409 0.87 HSD11B1 (0.47) CA12CA9RAB9ASMN1; SMN2CA1
SCHEMBL8079204 0.85 CNR2 (0.47) ALDH1A1CA12CA9NPC1RAB9A
SCHEMBL8092540 0.82 TAS2R14 (0.50) ALDH1A1NPC1RAB9ABMP1
SCHEMBL8079261 0.80 HSD11B1 (0.45) CA12CA9KCNH2KMT2AMEN1
SCHEMBL8090675 0.75 TAAR1 (0.43) CA12CA9RAB9ASMN1; SMN2TAAR1
SCHEMBL8092470 0.75 TAS2R14 (0.49) BMP1
SCHEMBL8087752 0.74 CES2 (0.43) CA12CA9NPC1RAB9ASMN1; SMN2
SCHEMBL8087638 0.74 TAS2R14 (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL8087708 0.74 TRPM8 (0.45) ALDH1A1RAB9ASMN1; SMN2KCNH2KMT2A
SCHEMBL6806990 0.74 PKM (0.52) ALDH1A1CA12CA9SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047670-A1 AMINOSULPHONYLBENZAMIDE DERIVATIVES AS MODULATORS OF THE ACTIVITY OF NEURONAL CALCIUM CHANNELS ELI LILLY AND COMPANY LIMITED (GB) 2000-11-02 EP disclosed
WO-1999036398-A1 AMINOSULPHONYLBENZAMIDE DERIVATIVES AS MODULATORS OF THE ACTIVITY OF NEURONAL CALCIUM CHANNELS ELI LILLY AND COMPANY LIMITED (GB) 1999-07-22 WO disclosed