SCHEMBL8090727

SCHEMBL8090727

CCCN(CCC)S(=O)(=O)N(Cc1cccc(C(F)(F)F)c1)C(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.51
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PDK1 Q15118 1/20 0.45
HSD11B1 P28845 1/20 0.43
PTGES O14684 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
CETP P11597 1/20 0.42
RAB9A P51151 1/20 0.41
NR3C1 P04150 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 2/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8087708 0.90 TRPM8 (0.45) TRPM8MEN1KMT2ALMNASMN1; SMN2
SCHEMBL8090715 0.84 TAS2R14 (0.53) MEN1KMT2ALMNAHSD11B1PTGES
SCHEMBL8087753 0.81 TAS2R14 (0.55) HSD11B1PTGES
SCHEMBL8087638 0.78 TAS2R14 (0.50) LMNASMN1; SMN2HSD11B1HDAC6RAB9A
SCHEMBL8092409 0.76 HSD11B1 (0.47) SMN1; SMN2HSD11B1HDAC6RAB9A
SCHEMBL8079261 0.74 HSD11B1 (0.45) MEN1KMT2ALMNAHSD11B1HDAC6
SCHEMBL8090718 0.73 TAS2R14 (0.47) SMN1; SMN2HSD11B1HDAC6RAB9AALDH1A1
SCHEMBL8087612 0.73 LPAR1 (0.43) MEN1KMT2ASMN1; SMN2HSD11B1ALDH1A1
SCHEMBL8086467 0.72 TAS2R14 (0.46) MEN1KMT2ASMN1; SMN2HSD11B1HDAC6
SCHEMBL8092470 0.72 TAS2R14 (0.49) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047670-A1 AMINOSULPHONYLBENZAMIDE DERIVATIVES AS MODULATORS OF THE ACTIVITY OF NEURONAL CALCIUM CHANNELS ELI LILLY AND COMPANY LIMITED (GB) 2000-11-02 EP disclosed
WO-1999036398-A1 AMINOSULPHONYLBENZAMIDE DERIVATIVES AS MODULATORS OF THE ACTIVITY OF NEURONAL CALCIUM CHANNELS ELI LILLY AND COMPANY LIMITED (GB) 1999-07-22 WO disclosed