SCHEMBL8094494

SCHEMBL8094494

Cc1nsc(NC(=O)Cc2cccc(Oc3ccc(N)cc3)c2)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 3/20 0.44
ALDH1A1 P00352 2/20 0.44
RAB9A P51151 1/20 0.44
CSNK1D P48730 3/20 0.40
PRKACA P17612 4/20 0.40
ROCK1 Q13464 4/20 0.40
P2RX4 Q99571 1/20 0.39
BRAF P15056 1/20 0.39
CYP3A4 P08684 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
RORC P51449 1/20 0.38
GLS O94925 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094492 0.90 MAPK8 (0.41) MAPK8ALDH1A1GLS
SCHEMBL7998311 0.83 GLS (0.44) MAPK8ALDH1A1RAB9AMAPTGLS
SCHEMBL7994626 0.80 GLS (0.42) MAPK8ALDH1A1RAB9AMAPTGLS
SCHEMBL8069562 0.76 MAPK8 (0.47) MAPK8RAB9ALMNAMAPTRORC
SCHEMBL8104093 0.76 KMT2A (0.49) MAPK8ALDH1A1RAB9ALMNAMAPT
SCHEMBL7230936 0.76 GAA (0.47) MAPK8ALDH1A1CSNK1D
SCHEMBL8094581 0.75 SMN1; SMN2 (0.40) MAPK8ALDH1A1RAB9ALMNAMAPT
SCHEMBL7232438 0.72 GLS (0.43) MAPK8ALDH1A1RAB9AROCK1LMNA
SCHEMBL7997967 0.72 KDM4E (0.41) ALDH1A1RAB9ACSNK1DLMNAMAPT
SCHEMBL7996112 0.70 RAB9A (0.51) MAPK8ALDH1A1RAB9ACSNK1DLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991631-A1 SUBSTITUTED AMINOHETEROCYCLYLAMIDES Bayer Aktiengesellschaft (DE) 2000-04-12 EP disclosed
WO-1999000375-A1 SUBSTITUTED AMINOHETEROCYCLYLAMIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-01-07 WO disclosed