SCHEMBL8103433

SCHEMBL8103433

CCc1cc(Cc2cc(CC)c(NC(=O)N(C)O)c(CC)c2)cc(CC)c1NC(=O)N(C)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.35
ALDH1A1 P00352 4/20 0.34
MAPT P10636 3/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
ALOX15 P16050 2/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 1/20 0.31
HTT P42858 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PKM P14618 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
SCN5A Q14524 1/20 0.30
PLK1 P53350 1/20 0.30
SHBG P04278 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25314219 0.77 HTT (0.42) GAAALDH1A1MAPTHPGDLMNA
SCHEMBL12284735 0.75 GAA (0.50) GAAALDH1A1MAPTHPGDLMNA
SCHEMBL13129145 0.71 PTPN1 (0.45) GAAALDH1A1MAPTHPGDLMNA
SCHEMBL13129142 0.71 HPGD (0.50) ALDH1A1HPGDCYP2C19KDM4E
SCHEMBL9861529 0.71 SHBG (0.34) GAAHPGDLMNAHTTMEN1
SCHEMBL12285477 0.70 KDM4E (0.54) ALDH1A1MAPTHPGDLMNAALOX15
SCHEMBL12284575 0.70 LMNA (0.50) GAAALDH1A1LMNAHTTMEN1
SCHEMBL8107899 0.69 GAA (0.57) GAALMNATSHRMEN1KMT2A
SCHEMBL12285484 0.69 EPHX2 (0.53) GAAALDH1A1MAPTHPGDCYP2C19
SCHEMBL14864150 0.69 HPGD (0.49) GAAHPGDLMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028291-A1 BISHYDROXYUREAS AS INHIBITORS OF THE 5-LIPOXYGENASE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1999-06-10 WO claimed
US-6121323-A LIPOXYGENASE INHIBITOR 3M INNOVATIVE PROPERTIES COMPANY (US) 2000-09-19 US disclosed
WO-1999028291-A1 BISHYDROXYUREAS AS INHIBITORS OF THE 5-LIPOXYGENASE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1999-06-10 WO disclosed