SCHEMBL820893

SCHEMBL820893

CC(C)c1cccc(N(c2ccc(N(c3ccc(N)cc3)c3ccc(N)cc3)cc2)c2cccc(C(C)C)c2C(C)C)c1C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.44
ALDH1A1 P00352 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CYP1A2 P05177 2/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPK1 P28482 2/20 0.35
TSHR P16473 2/20 0.35
PSMD14 O00487 1/20 0.35
RECQL P46063 1/20 0.35
GFER P55789 1/20 0.35
TP53 P04637 1/20 0.34
ALOX15 P16050 1/20 0.34
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13377362 0.80 GABRA1 (0.38) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL820809 0.78 L3MBTL1 (0.51) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL14562915 0.78 CYP3A4 (0.47) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL6933727 0.77 CYP3A4 (0.57) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL7028664 0.71 GABRA1 (0.43) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL22748315 0.70 GABRA1 (0.46) CYP3A4CYP1A2TSHRGABRA1GABRG2
SCHEMBL29088787 0.70 GABRA1 (0.41) CYP3A4CYP1A2TSHRGABRA1GABRG2
SCHEMBL7671735 0.69 CA1 (0.44) CYP3A4ALDH1A1TDP1CYP1A2TSHR
SCHEMBL13377297 0.68 CA1 (0.40) CYP3A4ALDH1A1TDP1L3MBTL1CYP1A2
SCHEMBL66227 0.67 GABRA1 (0.57) CYP3A4L3MBTL1CYP1A2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110275783-A1 Nitro compound, amine compound and polyamide derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2011-11-10 US claimed
US-20110275781-A1 Nitro compound, amine compound, polyimide and polyimide copolymer derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2011-11-10 US claimed
US-8492508-B2 Nitro compound, amine compound, polyimide and polyimide copolymer derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2013-07-23 US disclosed
US-8367797-B2 Nitro compound, amine compound and polyamide derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2013-02-05 US disclosed
US-20110275783-A1 Nitro compound, amine compound and polyamide derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2011-11-10 US disclosed
US-20110275781-A1 Nitro compound, amine compound, polyimide and polyimide copolymer derived therefrom NATIONAL TAIWAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (TW) 2011-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275783-A1 Nitro compound, amine compound and polyamide derived therefrom NOS2, NOS1, NOS3 CYP3A4 1179/4885ALDH1A1 2358/4885TDP1 1336/4885
US-20110275781-A1 Nitro compound, amine compound, polyimide and polyimide copolymer derived therefrom THEM6, NOS2, NOS1 CYP3A4 1102/4885ALDH1A1 2644/4885TDP1 2136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.