SCHEMBL8317710

SCHEMBL8317710

CCCN(C(=O)CC)C1CCc2c([N+](=O)[O-])ccc(Cl)c2C1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 3/20 0.37
ALDH1A1 P00352 1/20 0.37
DRD2 P14416 5/20 0.37
DRD1 P21728 3/20 0.37
OPRM1 P35372 2/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631076 0.88 DRD2 (0.36) DRD2DRD1OPRM1HTR1A
SCHEMBL8311336 0.85 HTR2A (0.43) DRD2HTR1A
SCHEMBL8318446 0.84 HTR1A (0.48) DRD2DRD1HTR1A
SCHEMBL8312041 0.77 HTR1A (0.51) ALDH1A1DRD2HTR1A
SCHEMBL7445601 0.76 DRD2 (0.42) DRD2DRD1HTR1A
SCHEMBL12640603 0.72 HTR1A (0.43) ALDH1A1DRD2HTR1A
SCHEMBL8318624 0.71 HTR1A (0.44) DRD2HTR1A
SCHEMBL10639140 0.70 DRD2 (0.58) DRD2HTR1A
SCHEMBL7433347 0.69 PNMT (0.47)
Hydrochloric Acid SCHEMBL8632206 0.69 LMNA (0.37) DRD2OPRM1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0510068-B1 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS UPJOHN CO (US) 1999-04-14 EP disclosed
US-5650427-A ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1997-07-22 US disclosed
US-5461061-A Antidepressants WIKSTROM HAKAN V (NL) 1995-10-24 US disclosed
US-5288748-A Antidepressants THE UPJOHN COMPANY (US) 1994-02-22 US disclosed
EP-0510068-A1 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS PHARMACIA & UPJOHN COMPANY (US) 1992-10-28 EP disclosed
WO-1991011435-A2 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS THE UPJOHN COMPANY (US) 1991-08-08 WO disclosed