SCHEMBL8325473

SCHEMBL8325473

O=C(O)CCc1ccc(N(C(=O)c2ccccc2)N2CCNCC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 7/20 0.44
PPARG P37231 2/20 0.43
KEAP1 Q14145 1/20 0.43
SIGMAR1 Q99720 1/20 0.40
FFAR4 Q5NUL3 2/20 0.40
SRD5A2 P31213 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
OPRM1 P35372 3/20 0.38
OPRD1 P41143 3/20 0.38
ADRA1A P35348 2/20 0.38
ADRA1B P35368 2/20 0.38
OPRK1 P41145 2/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
PTGIR P43119 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL379431 0.84 SIGMAR1 (0.51) SIGMAR1OPRM1OPRD1OPRK1USP2
SCHEMBL7536787 0.84 FFAR1 (0.41) FFAR1KEAP1FFAR4ITGB3ITGA2B
SCHEMBL4299855 0.76 SIGMAR1 (0.42) SIGMAR1OPRM1OPRD1OPRK1USP2
SCHEMBL7538929 0.72 AOC3 (0.37) ITGB3ITGA2BALDH1A1
Phenyl Propionic Acid SCHEMBL5057672 0.72 KEAP1 (0.76) FFAR1KEAP1FFAR4ADRA1AALDH1A1
Hydrochloric Acid SCHEMBL7538675 0.71 FKBP1A (0.43) ALDH1A1TSHR
SCHEMBL2302994 0.70 ITGB3 (0.61) FFAR1KEAP1SIGMAR1FFAR4ITGB3
SCHEMBL10900445 0.70 KCNH2 (0.57) FFAR1KEAP1SIGMAR1ITGB3ITGA2B
SCHEMBL5717885 0.68 SIGMAR1 (0.45) SIGMAR1OPRM1OPRD1USP2ALDH1A1
SCHEMBL7544912 0.68 CYP4A11 (0.38) SIGMAR1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912175-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-09-08 EP disclosed
EP-0912175-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1999-05-06 EP disclosed
WO-1998000134-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-01-08 WO disclosed